Activation of SIRT1 by silibinin improved mitochondrial health and alleviated the oxidative damage in experimental diabetic neuropathy and high glucose-mediated neurotoxicity

Arch Physiol Biochem. 2024 Aug;130(4):420-436. doi: 10.1080/13813455.2022.2108454. Epub 2022 Aug 9.

Abstract

Background: Silibinin (SBN), a sirtuin 1 (SIRT1) activator, has been evaluated for its anti-inflammatory activity in many inflammatory diseases. However, its role in diabetes-induced peripheral neuropathy (DPN) remains unknown. The SIRT1 activation convalesces nerve functions by improving mitochondrial biogenesis and mitophagy.

Methods: DPN was induced by streptozotocin (STZ) at a dose of 55 mg/kg, i.p. in the male SD rats whereas neurotoxicity was induced in Neuro2A cells by 30 mM (high glucose) glucose. Neurobehavioural (nerve conduction velocity and nerve blood flow) western blot, immunohistochemistry, and immunocytochemistry were performed to evaluate the protein expression and their cellular localisation.

Results: Two-week SBN treatment improved neurobehavioural symptoms, SIRT1, PGC-1α, and TFAM expression in the sciatic nerve and HG insulted N2A cells. It has also maintained the mitophagy by up-regulating PARL, PINK1, PGAM5, LC3 level and provided antioxidant defence by upregulating Nrf2.

Conclusion: SBN has shown neuroprotective potential in DPN through SIRT1 activation and antioxidant mechanism.

Keywords: Nrf2; SIRT1; Silibinin; mitochondrial biogenesis; mitochondrial protease.

MeSH terms

  • Animals
  • Antioxidants / pharmacology
  • Diabetes Mellitus, Experimental* / drug therapy
  • Diabetes Mellitus, Experimental* / metabolism
  • Diabetic Neuropathies* / drug therapy
  • Diabetic Neuropathies* / metabolism
  • Diabetic Neuropathies* / pathology
  • Glucose* / metabolism
  • Male
  • Mice
  • Mitochondria* / drug effects
  • Mitochondria* / metabolism
  • Mitophagy / drug effects
  • NF-E2-Related Factor 2 / metabolism
  • Neuroprotective Agents / pharmacology
  • Neuroprotective Agents / therapeutic use
  • Oxidative Stress* / drug effects
  • Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha / genetics
  • Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha / metabolism
  • Rats
  • Rats, Sprague-Dawley*
  • Sciatic Nerve / drug effects
  • Sciatic Nerve / metabolism
  • Silybin* / pharmacology
  • Sirtuin 1* / genetics
  • Sirtuin 1* / metabolism
  • Transcription Factors

Substances

  • Sirtuin 1
  • Silybin
  • Sirt1 protein, rat
  • Glucose
  • Neuroprotective Agents
  • Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha
  • Ppargc1a protein, rat
  • Antioxidants
  • NF-E2-Related Factor 2
  • Tfam protein, rat
  • Transcription Factors