Metformin inhibits the pathogenic functions of AChR-specific B and Th17 cells by targeting miR-146a

Immunol Lett. 2022 Oct:250:29-40. doi: 10.1016/j.imlet.2022.09.002. Epub 2022 Sep 13.

Abstract

Myasthenia gravis (MG) is characterized by fatigable skeletal muscle weakness with a fluctuating and unpredictable disease course and is caused by circulating autoantibodies and pathological T helper cells. Regulation of B-cell function and the T-cell network may be a potential therapeutic strategy for MG. MicroRNAs (miRNAs) have emerged as potential biomarkers in immune disorders due to their critical roles in various immune cells and multiple inflammatory diseases. Aberrant miR-146a signal activation has been reported in autoimmune diseases, but a detailed exploration of the relationship between miR-146a and MG is still necessary. Using an experimental autoimmune myasthenia gravis (EAMG) rat model, we observed that miR-146a was highly expressed in the spleen but expressed at low levels in the thymus and lymph nodes in EAMG rats. Additionally, miR-146a expression in T and B cells was also quite different. EAMG-specific Th17 and Treg cells had lower miR-146a levels, while EAMG-specific B cells had higher miR-146a levels, indicating that targeted intervention against miR-146a might have diametrically opposite effects. Metformin, a drug that was recently demonstrated to alleviate EAMG, may rescue the functions of both Th17 cells and B cells by reversing the expression of miR-146a. We also investigated the downstream target genes of miR-146a in both T and B cells using bioinformatics screening and qPCR. Taken together, our study identifies a complex role of miR-146a in the EAMG rat model, suggesting that more caution should be paid in targeting miR-146a for the treatment of MG.

Keywords: EAMG; Metformin; T cells, B cells; miR-146a.

MeSH terms

  • Animals
  • Autoantibodies
  • B-Lymphocytes
  • Biomarkers
  • Metformin* / pharmacology
  • Metformin* / therapeutic use
  • MicroRNAs* / genetics
  • Myasthenia Gravis, Autoimmune, Experimental* / drug therapy
  • Myasthenia Gravis, Autoimmune, Experimental* / genetics
  • Rats
  • Receptors, Cholinergic / immunology*
  • Th17 Cells

Substances

  • Autoantibodies
  • Biomarkers
  • MicroRNAs
  • Receptors, Cholinergic
  • Metformin