Subtypes of muscarinic receptors in cultured explants of the hippocampus of the rat

Neuropharmacology. 1987 Jul;26(7B):1027-9. doi: 10.1016/0028-3908(87)90082-7.

Abstract

Using the tritiated, muscarinic antagonist quinuclidinyl benzilate ([3H]QNB) as a ligand, muscarinic receptors have been identified and characterized in intact, cultured explants of the hippocampus of the rat. Competition studies with scopolamine and oxotremorine indicated a certain heterogeneity in the population of muscarinic receptors, whereas atropine and pirenzepine competed with [3H]QNB in a manner consistent with only one binding site for these substances. Thus, the observed heterogenity does not fit in with the M1/M2 receptor concept. Extended studies, with the aim of determining to what extent these putative subtypes of receptors are functional, would be of interest.

MeSH terms

  • Animals
  • Binding, Competitive
  • Hippocampus / analysis*
  • Oxotremorine / metabolism
  • Quinuclidinyl Benzilate / metabolism
  • Rats
  • Rats, Inbred Strains
  • Receptors, Muscarinic / analysis*
  • Scopolamine / metabolism

Substances

  • Receptors, Muscarinic
  • Oxotremorine
  • Quinuclidinyl Benzilate
  • Scopolamine