Fluoxetine combined with swimming exercise synergistically reduces lipopolysaccharide-induced depressive-like behavior by normalizing the HPA axis and brain inflammation in mice

Pharmacol Biochem Behav. 2023 Nov:232:173640. doi: 10.1016/j.pbb.2023.173640. Epub 2023 Sep 21.

Abstract

Major depression disorder is a debilitating psychiatric disease affecting millions of people worldwide. This disorder is the leading cause of morbidity and mortality in high-income countries. Selective serotonin reuptake inhibitors such as fluoxetine are first-line drugs for treating depression-related disorders, but not all patients respond well to these antidepressants. This study aimed to evaluate whether fluoxetine combined with aerobic exercise can affect lipopolysaccharide (LPS)-induced depressive-like behavior, hypothalamic-pituitary-adrenal (HPA) axis dysregulation, and brain inflammation in mice. Male mice were exposed to fluoxetine, swimming exercise, or a combination of both and finally treated with LPS. We measured depression-related symptoms such as anhedonia, behavioral despair, weight gain, and food intake. Hormones (corticosterone and testosterone) and cytokines (IL-1β, IL-6, TNF-α, IL-10) were also measured in serum and brain (hippocampus and prefrontal cortex), respectively. The findings indicated that LPS induced anhedonia and behavioral despair and increased corticosterone, hippocampal IL-1β, TNF-α, and decreased testosterone and hippocampal IL-10 in mice. Fluoxetine and exercise separately reduced LPS-induced depressive-like behavior, while their combination synergistically reduced these symptoms in LPS-treated mice. We found fluoxetine alone increased food intake and body weight in LPS-treated mice. Fluoxetine and exercise combination reduced corticosterone, hippocampal TNF-α, and prefrontal IL-6 and TNF-α levels and increased testosterone and hippocampal and prefrontal IL-10 levels more effectively than fluoxetine alone in LPS-treated mice. This study suggests that swimming exercise combined with fluoxetine can affect depression-related behavior, HPA axis, and brain inflammation more effectively than when they are used separately.

Keywords: Cytokines; HPG; Hippocampus; Mice; Physical activity; Prefrontal cortex.

MeSH terms

  • Anhedonia / drug effects
  • Animals
  • Behavior, Animal / drug effects
  • Corticosterone / blood
  • Cytokines / metabolism
  • Depression* / chemically induced
  • Depression* / drug therapy
  • Depression* / metabolism
  • Encephalitis / chemically induced
  • Encephalitis / metabolism
  • Encephalitis / psychology
  • Fluoxetine* / pharmacology
  • Hippocampus / drug effects
  • Hippocampus / metabolism
  • Hypothalamo-Hypophyseal System* / drug effects
  • Hypothalamo-Hypophyseal System* / metabolism
  • Lipopolysaccharides* / pharmacology
  • Male
  • Mice
  • Neuroinflammatory Diseases / drug therapy
  • Physical Conditioning, Animal* / physiology
  • Pituitary-Adrenal System* / drug effects
  • Pituitary-Adrenal System* / metabolism
  • Swimming*

Substances

  • Fluoxetine
  • Lipopolysaccharides
  • Corticosterone
  • Cytokines