5-Hydroxytryptamine depresses depolarizing responses to GABA in the rat isolated vagus nerve

Eur J Pharmacol. 1986 Nov 19;131(2-3):297-300. doi: 10.1016/0014-2999(86)90587-x.

Abstract

Axons of the rat isolated cervical vagus nerve responded to gamma-aminobutyric acid (GABA) and 5-hydroxytryptamine (5-HT) with a readily reversible dose-dependent depolarization. Prior application of 5-HT at 2 or 30 microM equally depressed the depolarizing responses to GABA, shifting the GABA dose-response curve to the right and depressing the maximum; by contrast, responses to 5-HT were affected only by large doses of GABA (greater than 300 microM), and to a lesser degree. In addition, the fade in responses to high doses of GABA was also reduced in the presence of 5-HT. It is suggested that such all-or-none depressive actions may explain the blockade of GABA-induced responses by 5-HT observed in other tissues such as the guinea-pig ileum.

MeSH terms

  • Animals
  • Electric Stimulation
  • GABA Antagonists*
  • In Vitro Techniques
  • Male
  • Neuromuscular Depolarizing Agents / antagonists & inhibitors*
  • Rats
  • Rats, Inbred Strains
  • Serotonin / pharmacology*
  • Vagus Nerve / drug effects*

Substances

  • GABA Antagonists
  • Neuromuscular Depolarizing Agents
  • Serotonin