Selective alteration in high affinity agonist binding: a mechanism of beta-adrenergic receptor desensitization

Mol Pharmacol. 1979 Jul;16(1):10-20.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenylyl Cyclases / blood
  • Adrenergic beta-Agonists / metabolism*
  • Adrenergic beta-Antagonists / blood
  • Animals
  • Anura
  • Binding, Competitive
  • Dihydroalprenolol / blood
  • Erythrocyte Membrane / metabolism
  • Guanine Nucleotides / pharmacology
  • In Vitro Techniques
  • Indicators and Reagents / pharmacology
  • Isoproterenol / blood
  • Rana pipiens
  • Receptors, Adrenergic / metabolism*
  • Receptors, Adrenergic, beta / drug effects
  • Receptors, Adrenergic, beta / metabolism*
  • Time Factors

Substances

  • Adrenergic beta-Agonists
  • Adrenergic beta-Antagonists
  • Guanine Nucleotides
  • Indicators and Reagents
  • Receptors, Adrenergic
  • Receptors, Adrenergic, beta
  • Dihydroalprenolol
  • Adenylyl Cyclases
  • Isoproterenol