Abstract
Mycobacterium tuberculosis (MTB) is a pathogenic bacterium, belonging to the family Mycobacteriaceae, that causes tuberculosis (TB). Toxoplasma gondii macrophage migration inhibitory factor (TgMIF), a protein homolog of macrophage migration inhibitory factor, has been explored for its potential to modulate immune responses during MTB infections. We observed that TgMIF that interacts with CD74, antizyme inhibitor 1 (AZIN1), and signal transducer and activator of transcription 1 (STAT1) modulates endocytosis, restoration of mitochondrial function, and macrophage polarization, respectively. These interactions promote therapeutic efficacy in mice infected with MTB, thereby presenting a potential route to host-directed therapy development. Furthermore, TgMIF, in combination with first-line TB drugs, significantly inhibited drug-resistant MTB strains, including multidrug-resistant TB. These results demonstrate that TgMIF is potentially a multifaceted therapeutic agent against TB, acting through immune modulation, enhancement of mitochondrial function, and dependent on STAT1 and AZIN1 pathways.
Publication types
-
Research Support, Non-U.S. Gov't
MeSH terms
-
Animals
-
Anti-Bacterial Agents* / metabolism
-
Anti-Bacterial Agents* / pharmacology
-
Antigens, Differentiation, B-Lymphocyte / metabolism
-
Binding Sites
-
Carrier Proteins / genetics
-
Carrier Proteins / metabolism
-
Cell Line
-
Chemotactic Factors* / genetics
-
Chemotactic Factors* / metabolism
-
Chemotactic Factors* / pharmacology
-
Drug Resistance, Bacterial
-
Endocytosis / drug effects
-
Female
-
Histocompatibility Antigens Class II / metabolism
-
Humans
-
Lung Injury / etiology
-
Lung Injury / pathology
-
Male
-
Mice
-
Mice, Inbred C57BL
-
Mice, Knockout
-
Mitochondria / drug effects
-
Mitochondria / metabolism
-
Mycobacterium tuberculosis* / drug effects
-
Mycobacterium tuberculosis* / metabolism
-
Protein Binding
-
STAT1 Transcription Factor / genetics
-
STAT1 Transcription Factor / metabolism
-
Signal Transduction* / drug effects
-
Toxoplasma* / genetics
-
Toxoplasma* / metabolism
-
Tuberculosis* / drug therapy
-
Tuberculosis* / genetics
-
Tuberculosis* / metabolism
-
Tuberculosis* / pathology
Substances
-
macrophage migration enhancement factor
-
Chemotactic Factors
-
Anti-Bacterial Agents
-
STAT1 Transcription Factor
-
ornithine decarboxylase antizyme inhibitor
-
Carrier Proteins
-
invariant chain
-
Histocompatibility Antigens Class II
-
Antigens, Differentiation, B-Lymphocyte