Radical scavenging effect of skin delivery systems using Korean red ginseng extract and assessment of their biocompatibility with human primary dermal fibroblasts and HaCaT keratinocytes

Int J Pharm. 2025 Apr 15:674:125477. doi: 10.1016/j.ijpharm.2025.125477. Epub 2025 Mar 15.

Abstract

Korean red ginseng (KRG) extract is proposed for cosmetic use, but no data on biological effects of KRG-loaded vehicles exist. The study aimed to optimize new multi- and monophase vehicles for KRG extract delivery, assess their biocompatibility and evaluate their radical scavenging effect in vitro. Storage stability of oil-in-water nanoemulsions (NEs) and hydroalcoholic gels (2 % w/w KRG) was assessed over twelve weeks using dynamic light scattering, rheology and pH measurements. Release profiles of ginsenosides Rb1 (more hydrophilic) and Rg1 (moderately lipophilic) through a cellulose membrane were also investigated employing Franz diffusion cells. Antioxidant potential and biocompatibility were assessed via 2,2-diphenyl-1-picrylhydrazyl (DPPH) and cell viability assays. Vehicles remained stable over twelve weeks at 8 °C (NEs Dh stable, gel viscosity + 3.5 %). Diffusion studies showed higher release of Rg1 vs. Rb1 (7.10 vs. 1.39 µg/cm-2 after 28 h). KRG-formulations demonstrated good biocompatibility with primary human dermal fibroblasts and HaCaT keratinocytes (72-94 % viability). Radical scavenging capacity of KRG extract did not differ between pure and incorporated form and was lower than that of a Hypericum extract or ascorbic acid. Results render KRG-formulations a potentially promising alternative to conventional antioxidants used in daily products.

Keywords: DPPH; HaCaT keratinocytes; Hydrogel; Korean red ginseng extract; Nanoemulsion; Primary human dermal fibroblasts; Release studies.

MeSH terms

  • Administration, Cutaneous
  • Antioxidants / chemistry
  • Biphenyl Compounds / chemistry
  • Cell Survival / drug effects
  • Drug Delivery Systems
  • Drug Liberation
  • Emulsions
  • Fibroblasts* / drug effects
  • Free Radical Scavengers* / administration & dosage
  • Free Radical Scavengers* / chemistry
  • Free Radical Scavengers* / pharmacology
  • Ginsenosides* / administration & dosage
  • Ginsenosides* / chemistry
  • Ginsenosides* / pharmacology
  • HaCaT Cells
  • Humans
  • Keratinocytes* / drug effects
  • Panax* / chemistry
  • Picrates
  • Plant Extracts* / administration & dosage
  • Plant Extracts* / chemistry
  • Plant Extracts* / pharmacology
  • Skin / cytology
  • Skin / drug effects
  • Skin / metabolism

Substances

  • Plant Extracts
  • Ginsenosides
  • Free Radical Scavengers
  • Emulsions
  • ginsenoside Rb1
  • Antioxidants
  • 1,1-diphenyl-2-picrylhydrazyl
  • Biphenyl Compounds
  • Picrates