Lycorine Inhibits Influenza Virus Replication by Affecting Nascent Nucleoporin Nup93 Synthesis

Int J Mol Sci. 2025 Jun 3;26(11):5358. doi: 10.3390/ijms26115358.

Abstract

The influenza A virus (IAV) is a major cause of recurrent seasonal epidemics and global pandemics, posing a significant threat to public health. Although lycorine has demonstrated broad-spectrum antiviral activity, its specific mechanisms of action against IAV remain incompletely understood. In this study, we characterized the potent inhibitory effects of lycorine on seasonal and drug-resistant IAV subtypes (H1N1/H3N2) as well as the influenza B virus, showing its ability to suppress viral mRNA, viral titers, and M2 protein expression across multiple cell lines. Time-of-addition and time-course assays revealed that lycorine exerts multiphasic interference, and the critical late stage of the IAV life cycle aroused our interest to study this further. Mechanistically, we discovered that lycorine specifically interferes with the de novo synthesis of nucleoporin Nup93, thereby disrupting the nuclear export of viral nucleoprotein (NP). These findings not only establish lycorine as a promising broad-spectrum anti-influenza candidate but also provide new insights for developing host-targeted antiviral strategies.

Keywords: Nup93; antiviral activity; influenza A virus; lycorine.

MeSH terms

  • A549 Cells
  • Amaryllidaceae Alkaloids* / pharmacology
  • Animals
  • Antiviral Agents* / pharmacology
  • Cell Line
  • Dogs
  • Humans
  • Influenza A Virus, H1N1 Subtype / drug effects
  • Influenza A Virus, H1N1 Subtype / physiology
  • Influenza A Virus, H3N2 Subtype / drug effects
  • Influenza A Virus, H3N2 Subtype / physiology
  • Influenza A virus* / drug effects
  • Influenza A virus* / physiology
  • Influenza B virus / drug effects
  • Influenza B virus / physiology
  • Influenza, Human / drug therapy
  • Influenza, Human / virology
  • Madin Darby Canine Kidney Cells
  • Nuclear Pore Complex Proteins* / biosynthesis
  • Nuclear Pore Complex Proteins* / genetics
  • Nuclear Pore Complex Proteins* / metabolism
  • Phenanthridines* / pharmacology
  • Virus Replication* / drug effects

Substances

  • lycorine
  • Amaryllidaceae Alkaloids
  • Phenanthridines
  • Antiviral Agents
  • Nuclear Pore Complex Proteins