Direct Oral Anticoagulants in Valvular Diseases and Prosthetic Valves: Why Not?

Cardiovasc Drugs Ther. 2026 Apr;40(2):697-709. doi: 10.1007/s10557-025-07736-8. Epub 2025 Jun 20.

Abstract

Valvular heart disease (VHD) and atrial fibrillation (AF) often coexist and lead to a prothrombotic state that necessitates the use of anticoagulants for the prevention of thromboembolic events. Direct oral anticoagulants (DOACs) are a significant advancement in anticoagulation therapy for patients with AF and VHD, leading to comparable efficacy and improved safety outcomes compared to vitamin K antagonists (VKAs). However, their role in patients with severe mitral stenosis, mechanical heart valves, and rheumatic heart disease remains limited due to the lack of robust data from clinical trials. As such warfarin continues to be the anticoagulant of choice for these populations. For patients with bioprosthetic valves or following transcatheter aortic valve implantation (TAVI), DOACs may be a viable alternative, but individualized risk assessment is crucial. The EHRA classification provides a practical framework for the management of patients with AF, but there are still challenges in its clinical application due to mixed valvular pathologies and patient-specific factors. Clinicians must carefully weigh the risk of thromboembolic and bleeding events, consider the patients' preferences, and advise regular follow-up to optimize the treatment outcomes. Overall, while DOACs offer convenience and similar efficacy and safety compared to VKAs, VKAs remain the anticoagulant of choice for specific subgroups, underscoring the need for personalized approaches regarding anticoagulation therapy.

Keywords: Atrial fibrillation (AF); DOACs; Prosthetic valves; Valvular heart disease (VHD).

Publication types

  • Review

MeSH terms

  • Administration, Oral
  • Anticoagulants* / administration & dosage
  • Anticoagulants* / adverse effects
  • Atrial Fibrillation* / diagnosis
  • Atrial Fibrillation* / drug therapy
  • Bioprosthesis
  • Factor Xa Inhibitors* / administration & dosage
  • Factor Xa Inhibitors* / adverse effects
  • Heart Valve Diseases* / diagnosis
  • Heart Valve Diseases* / drug therapy
  • Heart Valve Diseases* / surgery
  • Heart Valve Prosthesis Implantation* / adverse effects
  • Heart Valve Prosthesis Implantation* / instrumentation
  • Heart Valve Prosthesis*
  • Hemorrhage / chemically induced
  • Humans
  • Risk Assessment
  • Risk Factors
  • Thromboembolism* / diagnosis
  • Thromboembolism* / etiology
  • Thromboembolism* / prevention & control
  • Transcatheter Aortic Valve Replacement* / adverse effects
  • Transcatheter Aortic Valve Replacement* / instrumentation
  • Treatment Outcome

Substances

  • Anticoagulants
  • Factor Xa Inhibitors