Ghrelin-induced neuronal NPY promotes brain metastasis in lung cancer patients with low BMI

Nat Commun. 2025 Jul 1;16(1):5608. doi: 10.1038/s41467-025-60730-4.

Abstract

Obesity is a known risk factor for many cancers, yet recent studies reveal a paradoxical association between low body mass index (BMI) and increased brain metastasis in lung cancer-referred to as the "obesity paradox," with unclear molecular mechanism(s). Here, we show a significantly higher incidence of brain metastasis in low-BMI lung cancer patients compared to those with high-BMI or other cancer brain metastasis in a pan-analysis of 7628 patients. Mechanistically, low BMI activates ghrelin-GHSR signaling, increasing neuronal neuropeptide Y (NPY) secretion, which promotes tumor metabolic reprogramming via NPY-Y5R, facilitating brain colonization. Elevated plasma ghrelin levels in cancer-free low-BMI subjects suggest its potential as a prognostic biomarker for predicting brain metastasis. Notably, targeting NPY-Y5R or reversing low BMI effectively suppresses brain metastasis, supporting its pro-metastatic role. These findings provide a strong rationale for developing targeted interventions to treat or prevent brain metastasis in lung cancer patients with low BMI.

MeSH terms

  • Aged
  • Animals
  • Body Mass Index
  • Brain Neoplasms* / metabolism
  • Brain Neoplasms* / secondary
  • Cell Line, Tumor
  • Female
  • Ghrelin* / blood
  • Ghrelin* / metabolism
  • Humans
  • Lung Neoplasms* / metabolism
  • Lung Neoplasms* / pathology
  • Male
  • Mice
  • Middle Aged
  • Neurons* / metabolism
  • Neuropeptide Y* / genetics
  • Neuropeptide Y* / metabolism
  • Obesity / complications
  • Obesity / metabolism
  • Receptors, Ghrelin / metabolism
  • Receptors, Neuropeptide Y / metabolism
  • Signal Transduction

Substances

  • Ghrelin
  • Neuropeptide Y
  • Receptors, Ghrelin
  • Receptors, Neuropeptide Y