Per- and polyfluoroalkyl substances (PFAS) toxicity and mitigation of adipogenic dysregulation in 3T3-L1 preadipocytes

Food Chem Toxicol. 2025 Oct:204:115649. doi: 10.1016/j.fct.2025.115649. Epub 2025 Jul 16.

Abstract

Obesity and metabolic disorders are rising global concerns, with one factor linked to per- and polyfluoroalkyl substances (PFAS), a class of persistent endocrine-disrupting chemicals that affect adipogenic pathways. While PFAS are known to promote terminal lipid accumulation in mature adipocytes, their effects during dynamic adipocyte differentiation, particularly at human-relevant doses and in mixtures, remain poorly understood. This study employed 3T3-L1 preadipocytes to assess PFAS toxicity and mitigation in cell viability, redox balance, mitochondrial integrity, lipid content, and gene expression during differentiation. Repeated, low-dose exposure to 0.1 μM PFAS (individual and mixture) time-dependently reduced cell viability through induced reactive oxygen and nitrogen species by 22-49 % and reduced mitochondrial membrane potential. The 2-4-fold increase in lipid accumulation, especially by PFOA, correlated with Pparγ activation by 47-86 % (r2 ≥ 0.98). PFAS also triggered pro-inflammatory cytokines (Tnfα, Il-6) and suppressed anti-inflammatory mediators (Tgfβ, Il-10, Il-4), suggesting interactions between adipogenic and inflammatory pathways. Importantly, montmorillonite clays amended with choline or chlorophyll at 0.001 % and 0.01 % dose-dependently mitigated these effects, supporting critical PFAS pathways. By integrating mechanistic toxicology with mitigation interventions, this work establishes PFAS adipogenic toxicity through oxidative, metabolic, and inflammatory pathways, and supports nutrient-amended clays as sorbents to reduce PFAS bioavailability and prevent toxicity pathways during adipocyte development.

Keywords: Adipogenesis; Adsorption; Endocrine disrupting chemicals; Mitochondria; Obesity; Oxidative stress; Pparγ.

MeSH terms

  • 3T3-L1 Cells
  • Adipocytes* / drug effects
  • Adipocytes* / metabolism
  • Adipogenesis* / drug effects
  • Animals
  • Cell Differentiation / drug effects
  • Cell Survival / drug effects
  • Cytokines / metabolism
  • Fluorocarbons* / toxicity
  • Lipid Metabolism / drug effects
  • Membrane Potential, Mitochondrial / drug effects
  • Mice
  • Reactive Oxygen Species / metabolism

Substances

  • Fluorocarbons
  • Reactive Oxygen Species
  • Cytokines