Metabolism-dependent succinylation governs resource allocation for antibiotic resistance

Sci Adv. 2025 Aug 22;11(34):eadu2856. doi: 10.1126/sciadv.adu2856. Epub 2025 Aug 22.

Abstract

The mechanisms that organisms allocate resources to sustain biological phenotypes remain largely unknown. Here, we use mobilized colistin resistance (mcr-1), which modifies lipopolysaccharide (LPS) to confer colistin resistance, as a model to explore how bacteria reallocate resources to support mcr-1-mediated resistance. We show that bacteria redirect resources from glycolysis, the pyruvate cycle, and LPS biosynthesis toward glycerophospholipid metabolism to produce phosphatidylethanolamine, the substrate for mcr-1 to modify LPS, while reducing LPS content to limit colistin binding. This reallocation down-regulates succinyl-coenzyme A (CoA) to diminish succinylation of proteins including triosephosphate isomerase (TPI), CpxR, and PdhR, thereby sustaining resistance. Exogenous succinate or α-ketoglutarate restores succinylation in a succinyl-CoA-dependent manner. Succinylation of TPI redirects metabolic flux to glycolysis and the pyruvate cycle, while succinylation of CpxR and PdhR up-regulates LPS biosynthesis, ultimately attenuating colistin resistance. Thus, we reveal a previously unrecognized mechanism by which bacteria regulate resource allocation through metabolism-driven posttranslational protein modification, offering strategies to combat antibiotic resistance.

MeSH terms

  • Bacterial Proteins / metabolism
  • Colistin* / pharmacology
  • Down-Regulation
  • Drug Resistance, Bacterial*
  • Enterococcus faecalis* / drug effects
  • Enterococcus faecalis* / metabolism
  • Glycerophospholipids / metabolism
  • Glycolysis
  • Lipopolysaccharides / biosynthesis
  • Phosphatidylethanolamines / metabolism
  • Protein Processing, Post-Translational*
  • Triose-Phosphate Isomerase / metabolism
  • Up-Regulation

Substances

  • Colistin
  • Glycerophospholipids
  • Lipopolysaccharides
  • phosphatidylethanolamine
  • Phosphatidylethanolamines
  • CpxR protein, Bacteria
  • Bacterial Proteins
  • Triose-Phosphate Isomerase