Identification of Targetable EGFR Mutations in Ovarian Cancer

JCO Precis Oncol. 2025 Sep:9:e2500390. doi: 10.1200/PO-25-00390. Epub 2025 Sep 10.

Abstract

Purpose: EGFR mutations are classically seen in non-small cell lung cancers (NSCLCs), and EGFR-directed inhibitors have changed the therapeutic landscape in patients with EGFR-mutated NSCLC. The real-world prevalence of EGFR-mutated ovarian cancers has not been previously described. We aim to determine the prevalence of pathogenic or likely pathogenic EGFR mutations in ovarian cancer and describe a case of EGFR-mutated metastatic ovarian cancer with a durable response to osimertinib, an EGFR-directed targeted therapy.

Methods: Retrospective review of 33,850 molecularly profiled ovarian cancer samples from real-world patients who underwent next-generation sequencing (NGS) of DNA between 2016 and 2025. EGFR-mutated cases were defined as those harboring known pathogenic or likely pathogenic mutations based on the EGFR genomic alteration discovered by Caris.

Results: Of 33,850 patients, 27 (0.08%) harbored a genomic alteration in the EGFR gene that was pathogenic or likely pathogenic, including EGFR exon 20 mutation (n = 12, including five patients with EGFR T790M mutation), EGFR L858R (n = 3), and an EGFR exon 19 deletion (n = 2). Only one patient was treated with osimertinib, a third-generation EGFR-inhibitor, and achieved a durable objective response for over 17 months.

Conclusion: Ovarian cancer driven by an oncogenic EGFR mutation is a rare occurrence, yet it is an actionable molecular target with EGFR-directed inhibitors. This underlies the potential value of comprehensive NGS in the management of ovarian cancer for discovering actionable genomic alterations.

MeSH terms

  • Acrylamides / therapeutic use
  • Adult
  • Aged
  • Aged, 80 and over
  • Aniline Compounds / therapeutic use
  • ErbB Receptors* / genetics
  • Female
  • High-Throughput Nucleotide Sequencing
  • Humans
  • Indoles
  • Middle Aged
  • Mutation*
  • Ovarian Neoplasms* / drug therapy
  • Ovarian Neoplasms* / genetics
  • Protein Kinase Inhibitors / therapeutic use
  • Pyrimidines
  • Retrospective Studies

Substances

  • Acrylamides
  • Aniline Compounds
  • EGFR protein, human
  • ErbB Receptors
  • osimertinib
  • Protein Kinase Inhibitors
  • Indoles
  • Pyrimidines