Hybrid Exosome-Liposome Nanoparticles for Dual Modulation of Neuroinflammation and Lipid Metabolism in Ischemic Stroke

ACS Nano. 2025 Sep 23;19(37):33567-33586. doi: 10.1021/acsnano.5c11417. Epub 2025 Sep 15.

Abstract

Ischemic stroke, often modeled by middle cerebral artery occlusion and reperfusion (MCAO/R), involves severe neuroinflammation and lipid metabolic dysregulation that exacerbate neuronal damage. To address these dual pathological processes, we engineered a hybrid nanoplatform (Exo-Lip) by fusing neural stem cell-derived exosomes (Exo) with liposomes loaded with Yulangsan polysaccharide (Lip). Exosomes provide blood-brain barrier (BBB) permeability and intrinsic anti-inflammatory activity, while liposomes confer antioxidant and immunoregulatory effects. The resulting Exo-Lip exhibited improved colloidal stability and synergistic therapeutic potential. In MCAO/R mice, Exo-Lip markedly attenuated neuroinflammation by decreasing TNF-α and IL-6 while upregulating IL-10 and TGF-β. It restored lipid metabolism, alleviated oxidative stress, and preserved membrane integrity. TTC staining revealed a reduced infarct volume, and behavioral testing confirmed the recovery of motor and cognitive functions. Histological analyses further demonstrated neuronal survival and structural preservation. Transcriptomic profiling revealed that Exo-Lip modulated gene networks associated with inflammation and lipid regulation, including activation of the AKT/Nrf2/HO-1 signaling pathway. Collectively, these findings suggest that Exo-Lip represents a multifunctional, biomimetic nanotherapeutic capable of targeting both inflammatory and metabolic pathways in ischemic stroke. This work highlights a precision nanomedicine strategy with translational potential for central nervous system disorders.

Keywords: exosomes; ischemic stroke; lipid metabolism; liposomes; neuroinflammation.

MeSH terms

  • Animals
  • Exosomes* / chemistry
  • Exosomes* / metabolism
  • Inflammation / drug therapy
  • Ischemic Stroke* / drug therapy
  • Ischemic Stroke* / metabolism
  • Ischemic Stroke* / pathology
  • Lipid Metabolism* / drug effects
  • Liposomes* / chemistry
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Nanoparticles* / chemistry
  • Neuroinflammatory Diseases* / drug therapy
  • Neuroinflammatory Diseases* / metabolism

Substances

  • Liposomes