USP14-mediated metabolic competition impairs CD8+ T cell immunosurveillance in hepatocellular carcinoma

Proc Natl Acad Sci U S A. 2025 Sep 23;122(38):e2510576122. doi: 10.1073/pnas.2510576122. Epub 2025 Sep 18.

Abstract

Hepatocellular carcinoma (HCC) frequently develops resistance to CD8+ T cell-based immunotherapy, yet the mechanisms driving this immune evasion remain poorly understood. To identify tumor-intrinsic regulators of immunotherapy resistance and explore therapeutic strategies to restore T cell-mediated tumor control, we employed three functional genomics approaches using in vitro and in vivo CRISPR screening. Cancer USP14 was identified as the critical immune evasion driver. USP14-high HCC patients exhibited poorer anti-PD1 antibody therapy responses and reduced CD8+ T cell infiltration. Inhibition of USP14 suppressed HCC cell growth in coculture with activated CD8+ T cells and restored cocultured CD8+ T cell cytotoxicity. In vivo USP14 targeting synergized with anti-PD1 antibody therapy. Mechanistically, USP14 deubiquitinated and stabilized GLUT1 through the removal of Lys-48-linked ubiquitin chains at Lys-245, which enabled HCC cells to outcompete CD8+ T cells for glucose, generating a glucose-deprived tumor microenvironment that suppressed CD8+ T cell function. Our findings show USP14 in cancer has a proimmunoevasive role in CD8+ T cell-based tumor immunity through GLUT1-mediated glucose competition. These findings position USP14 inhibitors as promising adjuvants to enhance immunotherapy efficacy in HCC, providing actionable insights for overcoming resistance.

Keywords: GLUT1; USP14; glucose competition; hepatocellular carcinoma.

MeSH terms

  • Animals
  • CD8-Positive T-Lymphocytes* / immunology
  • CD8-Positive T-Lymphocytes* / metabolism
  • Carcinoma, Hepatocellular* / genetics
  • Carcinoma, Hepatocellular* / immunology
  • Carcinoma, Hepatocellular* / metabolism
  • Carcinoma, Hepatocellular* / pathology
  • Cell Line, Tumor
  • Glucose / metabolism
  • Glucose Transporter Type 1 / metabolism
  • Humans
  • Immunologic Surveillance*
  • Immunotherapy
  • Liver Neoplasms* / genetics
  • Liver Neoplasms* / immunology
  • Liver Neoplasms* / metabolism
  • Liver Neoplasms* / pathology
  • Mice
  • Programmed Cell Death 1 Receptor / antagonists & inhibitors
  • Programmed Cell Death 1 Receptor / immunology
  • Tumor Microenvironment / immunology
  • Ubiquitin Thiolesterase* / genetics
  • Ubiquitin Thiolesterase* / immunology
  • Ubiquitin Thiolesterase* / metabolism

Substances

  • Ubiquitin Thiolesterase
  • Glucose Transporter Type 1
  • SLC2A1 protein, human
  • Programmed Cell Death 1 Receptor
  • Glucose