Brief Primer on the Discovery of New Antifungal Drugs from Plant Sources

Mycopathologia. 2025 Oct 11;190(6):102. doi: 10.1007/s11046-025-01009-6.

Abstract

Rationale: The antifungal armamentarium is shrinking while resistance to licensed agents rises. Historically, actinomycetes and fungi delivered nystatin, amphotericin B, griseofulvin and the echinocandin scaffold, yet plant-derived compounds-despite potent in-vitro activity-have rarely reached the clinic.

Objective: To frame the recent in-vivo success of papaya-seed essential oil against fluconazole-sensitive and -resistant Candida albicans within the broader context of plant-based antifungal discovery, and to propose rigorous criteria that can accelerate translation, especially considering varying resource settings.

Key points: Commentary on Ma et al. (Mycopathologia 190(5):1-14, 2025) showing that benzyl-isothiocyanate-rich papaya-seed oil outperforms fluconazole in a murine systemic candidiasis model without acute toxicity; Historical perspective on how soil microbes provided the first broad-spectrum antifungals; An eight-point checklist for future plant-extract studies, with essential and suggested elements to promote high-quality research across different laboratory settings.

Conclusion: Adherence to core methodological standards, along with suggested advanced analyses where feasible, will help identify promising plant-derived antifungal leads and support a more inclusive and effective discovery pipeline.

Keywords: Candida albicans; Benzyl isothiocyanate; Drug resistance; Plant antifungals; Translational research.

Publication types

  • Review
  • Letter

MeSH terms

  • Animals
  • Antifungal Agents* / isolation & purification
  • Antifungal Agents* / pharmacology
  • Antifungal Agents* / therapeutic use
  • Candida albicans* / drug effects
  • Candidiasis / drug therapy
  • Disease Models, Animal
  • Drug Discovery* / methods
  • Drug Resistance, Fungal
  • Humans
  • Mice
  • Microbial Sensitivity Tests
  • Oils, Volatile / isolation & purification
  • Oils, Volatile / pharmacology
  • Plant Extracts* / pharmacology
  • Plants* / chemistry

Substances

  • Antifungal Agents
  • Plant Extracts
  • Oils, Volatile