Integrative mapping reveals molecular features underlying the mechanism of nucleocytoplasmic transport

Proc Natl Acad Sci U S A. 2025 Oct 21;122(42):e2507559122. doi: 10.1073/pnas.2507559122. Epub 2025 Oct 16.

Abstract

Nuclear pore complexes (NPCs) enable rapid, selective, and robust nucleocytoplasmic transport. To explain how transport emerges from the system components and their interactions, we used experimental data and theoretical information to construct an integrative Brownian dynamics model of transport through an NPC, coupled to a kinetic model of transport in the cell. The model recapitulates key aspects of transport for a wide range of molecular cargoes, including preribosomes and viral capsids. Our model quantifies how flexible phenylalanine-glycine (FG) repeat proteins create an entropic barrier to passive diffusion and how this barrier is selectively lowered in facilitated diffusion by the many transient interactions of nuclear transport receptors with the FG repeats. Selective transport is enhanced by "fuzzy" multivalent interactions, redundant FG repeat mass, coupling to the energy-dependent RanGTP concentration gradient, and exponential dependence of transport kinetics on the transport barrier. Our model will facilitate rational modulation of the NPC and its artificial mimics.

Keywords: Brownian dynamics simulations; integrative modeling; nuclear pore complex; nucleocytoplasmic transport; spatiotemporal modeling.

MeSH terms

  • Active Transport, Cell Nucleus* / physiology
  • Diffusion
  • Kinetics
  • Models, Biological*
  • Nuclear Pore Complex Proteins / metabolism
  • Nuclear Pore* / metabolism
  • ran GTP-Binding Protein / metabolism

Substances

  • Nuclear Pore Complex Proteins
  • ran GTP-Binding Protein