Bictegravir/emtricitabine/tenofovir alafenamide for primary HIV infection: Efficacy, safety and impact on viral reservoir (the BIC-PHI clinical trial)

J Infect. 2025 Nov;91(5):106651. doi: 10.1016/j.jinf.2025.106651. Epub 2025 Nov 7.

Abstract

Objectives: We evaluated the efficacy, safety and impact on viral reservoir of rapid bictegravir/emtricitabine/tenofovir alafenamide (BIC/FTC/TAF) initiation during primary HIV infection (PHI).

Methods: Multicenter, single-arm clinical trial in participants with PHI of <3 months (seroconversion or incomplete serological pattern), starting BIC/FTC/TAF in 6 Spanish centers between January-2021 and September-2022. Primary endpoint was proportion of participants with viral load (VL)<50 copies/mL at 48-weeks on the Intention-to-treat-exposed population (ITTe). Cases were compared with randomly-matched retrospective PHI controls, starting other 3-drug Integrase-Strand-Transfer-inhibitor-based regimens. Reservoir was evaluated in PHI cases by Intact Proviral DNA Assay (IPDA).

Results: We included 64 participants, 94% cis-male, aged 32 (26;41) years.; 78% men-who-have-sex-with-men. At BIC/FTC/TAF initiation, Fiebig stages were II (14%), III (11%); IV (5%), V (54%) and VI (16%); VL was 496,520 (110,000;1,285,000) copies/mL; 62% were subtype B; median (IQR) CD4 T cell count was 406 (322;535) cells/µL; 6% had active hepatitis B virus co-infection. All participants started BIC/FTC/TAF at first specialist consultation. 81% (ITTe) and 93% (On-Treatment, OT) had VL<50 copies/mL at 48-weeks. 72% had adverse events, only 3% were grade 3/4; 91% were not-related, none led to BIC/FTC/TAF-discontinuation. 92% of controls (OT) had VL<50 copies/mL at 48-weeks (p=0.914), 11% (17%) modified initial antiretroviral regimen (p>0.001). Intact and defective proviral DNA levels significantly decreased at 48-weeks.

Conclusions: BIC/FTC/TAF showed rapid viral decay, high suppression rates, good tolerability, and reservoir decline in PHI, making it an appealing regimen in this setting.

Keywords: BIC/FTC/TAF; Bictegravir; PHI; Primary HIV infection; Rapid ART initiation; Viral load; Viral reservoir; Viral suppression.

Publication types

  • Multicenter Study

MeSH terms

  • Adenine* / analogs & derivatives
  • Adenine* / therapeutic use
  • Adult
  • Alanine
  • Amides
  • Anti-HIV Agents* / adverse effects
  • Anti-HIV Agents* / therapeutic use
  • Drug Combinations
  • Emtricitabine* / adverse effects
  • Emtricitabine* / therapeutic use
  • Female
  • HIV Infections* / drug therapy
  • HIV Infections* / virology
  • HIV-1 / drug effects
  • Heterocyclic Compounds, 3-Ring / therapeutic use
  • Heterocyclic Compounds, 4 or More Rings* / therapeutic use
  • Humans
  • Male
  • Middle Aged
  • Piperazines / therapeutic use
  • Pyridones / therapeutic use
  • Spain
  • Tenofovir* / analogs & derivatives
  • Tenofovir* / therapeutic use
  • Treatment Outcome
  • Viral Load / drug effects

Substances

  • Emtricitabine
  • Tenofovir
  • Anti-HIV Agents
  • bictegravir
  • Pyridones
  • Adenine
  • Alanine
  • Heterocyclic Compounds, 4 or More Rings
  • Piperazines
  • tenofovir alafenamide
  • Heterocyclic Compounds, 3-Ring
  • Drug Combinations
  • Amides