Boric acid-functionalized bentonite nanostructures attenuated paraquat-induced pulmonary injuries in rats

Sci Rep. 2025 Dec 8;15(1):43321. doi: 10.1038/s41598-025-27334-w.

Abstract

This study evaluated the antioxidant, anti-inflammatory, and anti-fibrotic effects of boric acid-functionalized bentonite nanostructures (BABTs) in a rat model of paraquat (PQ)-induced pulmonary toxicity, a well-established model for herbicide-related lung fibrosis. BABTs (20-60 nm) were synthesized via a microwave-assisted technique, characterized by dynamic light scattering, scanning electron microscopy, Fourier-transform infrared, and ultraviolet-visible spectroscopy, confirming PQ-BABT complex formation. Forty-eight male Wistar rats were randomized into eight groups (n = 6/group): negative control (saline), positive control (single 100 mg/kg PQ oral dose), and experimental groups receiving BABTs or boric acid (BA) at 10, 50, or 100 mg/kg/day orally, 30 min post-PQ. After 14 days, lung malondialdehyde (MDA) levels and histopathological changes (H&E, Masson's Trichrome) were assessed. BABTs at 50 mg/kg significantly decreased lung malondialdehyde (MDA) levels (P < 0.05) and significantly attenuated tissue injury (P < 0.05), suggesting an attenuation of oxidative stress, inflammation, and fibrosis, while boric acid (BA) demonstrated no significant effect. BABTs mitigate PQ-induced lung injury through antioxidant, anti-inflammatory, and anti-fibrotic mechanisms, enhanced by reducing PQ bioavailability. These findings position BABTs as a promising therapeutic candidate for PQ-induced pulmonary fibrosis, warranting further clinical evaluation.

Keywords: Boric acid; Functionalized bentonite nanostructures; Paraquat; Pulmonary fibrosis; Rat.

MeSH terms

  • Animals
  • Antioxidants / chemistry
  • Antioxidants / pharmacology
  • Bentonite* / chemistry
  • Bentonite* / pharmacology
  • Boric Acids* / chemistry
  • Boric Acids* / pharmacology
  • Disease Models, Animal
  • Herbicides / toxicity
  • Lung / drug effects
  • Lung / metabolism
  • Lung / pathology
  • Lung Injury* / chemically induced
  • Lung Injury* / drug therapy
  • Lung Injury* / pathology
  • Male
  • Malondialdehyde / metabolism
  • Nanostructures* / chemistry
  • Oxidative Stress / drug effects
  • Paraquat* / toxicity
  • Pulmonary Fibrosis / chemically induced
  • Pulmonary Fibrosis / drug therapy
  • Pulmonary Fibrosis / pathology
  • Rats
  • Rats, Wistar

Substances

  • Boric Acids
  • Paraquat
  • boric acid
  • Bentonite
  • Antioxidants
  • Herbicides
  • Malondialdehyde