Enhanced insulin signaling via circulating ATG7: A potential therapeutic strategy for diabetes

Proc Natl Acad Sci U S A. 2026 Jan 6;123(1):e2503783123. doi: 10.1073/pnas.2503783123. Epub 2025 Dec 29.

Abstract

Diabetes and insulin resistance (IR) remain major global health challenges, underscoring the need for novel therapeutic strategies. Here, we identify an autophagy-independent role of circulating autophagy-related gene 7 (ATG7) in metabolic regulation. Circulating ATG7 enhances insulin sensitivity and glucose homeostasis by directly interacting with IRS1 and modulating insulin signaling (IS) through liver-muscle crosstalk. Mechanistically, ATG7 binds to IRS1, promoting its activation and the propagation of downstream IS. Notably, we identify an ATG7-derived peptide (Aap2) that recapitulates ATG7's insulin-sensitizing effects and improves glycemic control in both Type 1 and Type 2 diabetic mouse models. These findings establish ATG7 as a key regulator of IS and suggest that targeting ATG7 may represent a promising therapeutic approach for IR and diabetes.

Keywords: ATG7; IRS1; exosomes; glucose homeostasis; insulin resistance.

MeSH terms

  • Animals
  • Autophagy
  • Autophagy-Related Protein 7* / blood
  • Autophagy-Related Protein 7* / genetics
  • Autophagy-Related Protein 7* / metabolism
  • Diabetes Mellitus, Experimental / metabolism
  • Diabetes Mellitus, Type 1* / blood
  • Diabetes Mellitus, Type 1* / drug therapy
  • Diabetes Mellitus, Type 1* / metabolism
  • Diabetes Mellitus, Type 2* / blood
  • Diabetes Mellitus, Type 2* / drug therapy
  • Diabetes Mellitus, Type 2* / metabolism
  • Humans
  • Insulin Receptor Substrate Proteins / metabolism
  • Insulin Resistance
  • Insulin* / metabolism
  • Liver / metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Signal Transduction*

Substances

  • Insulin
  • Autophagy-Related Protein 7
  • Insulin Receptor Substrate Proteins
  • Atg7 protein, mouse
  • Irs1 protein, mouse