Site-specific HPV18 integration facilitates cervical carcinogenesis through metabolic reprogramming-induced dysfunction of the SpHK1/S1P/S1PR1 pathway

Cell Death Dis. 2026 Jan 9;17(1):24. doi: 10.1038/s41419-025-08195-7.

Abstract

Integration of high-risk human papillomavirus into specific loci of the genome is a pivotal event in cervical carcinogenesis; however, it's underlying mechanism remains largely undefined. Here, through establishing an 8q24 site-specific HPV18 gene knock-in cell model by utilizing the CRISPR/Cas9 system, we discover that HPV18 knock-in (HPV-KI) results in a global alteration of the genome's topologically associating domain structure and an up-regulation of cancer-related genes in HPV- HaCaT cells, among which the significantly up-regulated IL-17 signaling pathway and S100A8/A9 are partitularly prominent. Further mechanistic study demonstrate that HPV-KI reprograms metabolic pathway, especially up-regulates glycolysis and subsequently facilitates glycerolipid synthesis in HaCaT cell, leading to sphingosine-1-phospate (S1P) secretion and enhanced SpHK1/S1P/S1PR1 signaling pathway, thereby activating the the MAPK and NF-κB signaling pathways followed by inducing the expression of S100A8/A9, and hence induces the malignant transformation of cells. Importantly, inhibition of the S1P/S1PR1 signaling pathway down-regulates the expression of S100A8/A9 and suppresses the growth of HPV-KI cells and xenograft derived from cervical cancer patient. These findings provide novel insights into HPV integration-induced cervical carcinogenesis and identify potential therapeutic targets for its treatment.

MeSH terms

  • Animals
  • Calgranulin B / metabolism
  • Carcinogenesis* / genetics
  • Carcinogenesis* / metabolism
  • Carcinogenesis* / pathology
  • Female
  • HaCaT Cells
  • Human papillomavirus 18* / genetics
  • Humans
  • Metabolic Reprogramming
  • Mice
  • Mice, Nude
  • Papillomavirus Infections / virology
  • Phosphotransferases (Alcohol Group Acceptor)* / metabolism
  • Signal Transduction
  • Sphingosine Kinase
  • Sphingosine-1-Phosphate Receptors* / metabolism
  • Uterine Cervical Neoplasms* / genetics
  • Uterine Cervical Neoplasms* / metabolism
  • Uterine Cervical Neoplasms* / pathology
  • Uterine Cervical Neoplasms* / virology
  • Virus Integration*

Substances

  • Sphingosine-1-Phosphate Receptors
  • Phosphotransferases (Alcohol Group Acceptor)
  • Calgranulin B
  • Sphingosine Kinase
  • S1PR1 protein, human