Oral Centella asiatica Extract Attenuates UVB-Induced Skin Photoaging via Antioxidant, Anti-Inflammatory, and Extracellular Matrix-Preserving Effects in Hairless Mice

Int J Mol Sci. 2025 Dec 24;27(1):204. doi: 10.3390/ijms27010204.

Abstract

Centella asiatica exhibits antioxidant, anti-inflammatory, and dermal-regenerative activities, yet the in vivo efficacy of an orally administered, dose-standardized extract against ultraviolet B (UVB)-induced photoaging has not been fully elucidated. This study investigated the protective effects of a chemically standardized C. asiatica extract (sCAE; 70 mg/g asiaticoside) in UVB-irradiated Skh:HR-1 hairless mice. Animals received oral sCAE (40 or 80 mg/kg/day) for eight weeks during repeated UVB exposure. Comprehensive assessments-including skin biophysical measurements, histological analysis, ELISA, and gene expression profiling-were performed to characterize dose-dependent responses. sCAE significantly reduced wrinkle formation, transepidermal water loss, malondialdehyde accumulation, and pro-inflammatory cytokines, while enhancing skin hydration, elasticity, antioxidant enzyme activities, and collagen expression. It also restored hyaluronic acid, ceramide, and their biosynthetic genes, and suppressed matrix metalloproteinase-1 and -9. Notably, the higher dose (80 mg/kg) consistently shifted key parameters toward normal levels, demonstrating a clear dose-response effect. These findings provide the first integrative in vivo evidence that orally administered, asiaticoside-standardized C. asiatica extract mitigates UVB-induced photoaging by concurrently improving barrier lipids, extracellular matrix integrity, inflammation, and oxidative stress, supporting its potential as a nutricosmetic agent for skin health.

Keywords: Centella asiatica; UVB-induced photoaging; anti-inflammatory effect; antioxidant enzymes; collagen preservation; hairless mice; oral administration.

MeSH terms

  • Administration, Oral
  • Animals
  • Anti-Inflammatory Agents* / administration & dosage
  • Anti-Inflammatory Agents* / pharmacology
  • Antioxidants* / administration & dosage
  • Antioxidants* / pharmacology
  • Centella / chemistry
  • Extracellular Matrix* / drug effects
  • Extracellular Matrix* / metabolism
  • Female
  • Mice
  • Mice, Hairless
  • Plant Extracts / pharmacology
  • Skin / drug effects
  • Skin / metabolism
  • Skin / radiation effects
  • Skin Aging* / drug effects
  • Skin Aging* / radiation effects
  • Triterpenes* / administration & dosage
  • Triterpenes* / pharmacology
  • Ultraviolet Rays* / adverse effects

Substances

  • Antioxidants
  • Centella asiatica extract
  • Anti-Inflammatory Agents
  • Triterpenes
  • Plant Extracts