CXCL9 and CXCL10 Induce Expression of Nociceptive Ion Channels in Primary Sensory Neurons in Models of HIV-Associated Distal Sensory Polyneuropathy

Int J Mol Sci. 2026 Jan 4;27(1):523. doi: 10.3390/ijms27010523.

Abstract

HIV-associated distal sensory polyneuropathy (HIV-DSP) remains prevalent even in the antiretroviral therapy (ART) era. Previously, we identified the upregulation of nociceptive ion channels transient receptor potential vanilloid 1 (TRPV1) and ankyrin 1 (TRPA1) in the dorsal root ganglia (DRG) of simian immunodeficiency virus (SIV)-infected ART-treated macaques. To investigate upstream mechanisms, we performed bulk RNA-seq and pathway analysis on DRGs from uninfected, SIV-infected, and SIV-infected/ART macaques. SIV infection drove strong activation of upstream regulators of interferon γ (IFNγ) and lipopolysaccharide (LPS). Although ART reduced overall IFNγ and LPS pathway activity, the IFNγ-inducible chemokines C-X-C motif chemokine ligand (CXCL)9 and CXCL10 remained significantly upregulated. To determine whether these chemokines influence TRPV1/TRPA1 expression, we treated induced pluripotent stem cell-derived peripheral sensory neurons (iPSC-PSNs) with CXCL9 and CXCL10, which induced a significant increase in TRPV1 but not TRPA1 expression. In parallel experiments, IFNγ but not LPS stimulated monocyte-derived macrophages (MDMs) to release CXCL9 and CXCL10. Conditioned media from IFNγ-treated MDMs modestly increased TRPV1 expression in iPSC-PSNs, and pharmacological inhibition of CXCR3, the receptor of CXCL9/10, did not reduce this effect. Together, these data indicate that persistent IFNγ-driven CXCL9/10 signaling may be one contributor to nociceptor sensitization underlying HIV-DSP, even in the presence of ART.

Keywords: HIV; SIV; neuroinflammation; neuropathy.

MeSH terms

  • Animals
  • Ankyrins* / metabolism
  • Anti-Retroviral Agents / therapeutic use
  • Chemokine CXCL10 / metabolism
  • Chemokine CXCL9 / metabolism
  • Ganglia, Spinal* / metabolism
  • Humans
  • Macaca mulatta
  • Nociceptors* / metabolism
  • Polyneuropathies* / metabolism
  • Polyneuropathies* / virology
  • Simian Acquired Immunodeficiency Syndrome / complications
  • Simian Acquired Immunodeficiency Syndrome / drug therapy
  • TRPV Cation Channels* / metabolism
  • Transcriptome

Substances

  • Chemokine CXCL9
  • Chemokine CXCL10
  • Anti-Retroviral Agents
  • TRPV1 receptor
  • TRPV Cation Channels
  • Ankyrins