Maresin 1 ameliorates myocardial ischaemia‒reperfusion injury by promoting tissue resident macrophage efferocytosis

Cardiovasc Res. 2026 Mar 26;122(3):397-411. doi: 10.1093/cvr/cvag017.

Abstract

Aims: Myocardial ischaemia‒reperfusion (I/R) injury triggers a robust inflammatory storm cascade that critically compromises reperfusion efficacy following acute myocardial infarction. Enhanced efferocytosis by cardiac resident macrophages (RMs) has therapeutic potential for inflammation resolution. The unsaturated long-chain fatty acid Maresin1 (MaR1) exhibits potent anti-inflammatory properties that is devoid of immunosuppressive effects. However, its therapeutic potential in myocardial I/R injury and regulatory mechanisms in cardiac RMs remains unexplored.

Methods and results: A clinical case‒control study was conducted and revealed a negative association between circulating MaR1 levels and inflammatory markers and the severity of I/R injury in patients with ST-elevation myocardial infarction. Mice treated with MaR1 after myocardial I/R injury showed improvements in cardiac function and efferocytosis by cardiac RMs. Genetic ablation of cardiac RMs abolished MaR1-mediated cardioprotection. To explore the mechanism underlying this protection, we performed transcriptomic, metabolomics, and lipidomic analyses and identified fatty acid β-oxidation potentiation as a key metabolic signature in MaR1-treated RMs. Moreover, MaR1 directly bound peroxisome proliferator-activated receptor γ (PPARγ), inducing the transcriptional activation of its downstream efferocytosis-related target CD204. Specific knockout of PPARγ in RMs significantly attenuated MaR1-enhanced efferocytosis. Notably, oral supplementation with the MaR1 precursor docosahexaenoic acid (DHA) recapitulated these cardioprotective effects.

Conclusion: Our findings prove that MaR1 plays a protective role in myocardial I/R injury by facilitating efferocytosis by RMs and the resolution of inflammation. These results offer novel therapeutic perspectives for the management of myocardial I/R injury.

Keywords: Efferocytosis; Inflammation; Maresin 1; Myocardial I/R injury; Resident macrophage.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents* / pharmacology
  • Case-Control Studies
  • Disease Models, Animal
  • Docosahexaenoic Acids* / pharmacology
  • Efferocytosis
  • Female
  • Humans
  • Inflammation Mediators / blood
  • Inflammation Mediators / metabolism
  • Macrophages* / drug effects
  • Macrophages* / metabolism
  • Macrophages* / pathology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Middle Aged
  • Myocardial Reperfusion Injury* / genetics
  • Myocardial Reperfusion Injury* / metabolism
  • Myocardial Reperfusion Injury* / pathology
  • Myocardial Reperfusion Injury* / physiopathology
  • Myocardial Reperfusion Injury* / prevention & control
  • Myocardium* / metabolism
  • Myocardium* / pathology
  • PPAR gamma / genetics
  • PPAR gamma / metabolism
  • Phagocytosis* / drug effects
  • ST Elevation Myocardial Infarction* / drug therapy
  • ST Elevation Myocardial Infarction* / genetics
  • ST Elevation Myocardial Infarction* / metabolism
  • ST Elevation Myocardial Infarction* / pathology
  • ST Elevation Myocardial Infarction* / physiopathology
  • Signal Transduction
  • Ventricular Function, Left / drug effects

Substances

  • Docosahexaenoic Acids
  • 7,14-dihydroxydocosa-4,8,10,12,16,19-hexaenoic acid
  • PPAR gamma
  • Anti-Inflammatory Agents
  • Inflammation Mediators
  • Pparg protein, mouse