PCIF1 Attenuates Type I Interferon Induction by Inhibiting IRF3 Activation in a Methyltransferase-Independent Manner

Cells. 2026 Feb 5;15(3):303. doi: 10.3390/cells15030303.

Abstract

PCIF1 is primarily recognized as an RNA methyltransferase that mediates N6-methylation of cap-proximal adenosine (m6Am) and plays diverse roles in gene expression. In this study, we uncover a novel role for PCIF1 as a crucial negative regulator of type I interferon (IFN) induction, a pathway critical for antiviral immunity whose dysregulation leads to inflammatory and autoimmune diseases. We demonstrate that PCIF1 deficiency robustly enhances the poly(I:C)-induced type I IFN response, accompanied by augmented STAT1 activation and interferon-stimulated gene (ISG) expression. Mechanistically, PCIF1 suppresses IFNB1 transcription by attenuating IRF3 phosphorylation and nuclear translocation, as shown by increased nascent IFNB1 mRNA synthesis and promoter activity in PCIF1-deficient cells, without affecting the mRNA stability. Crucially, this suppressive function was independent of PCIF1's canonical RNA methyltransferase activity, as both wild-type PCIF1 and a methyltransferase-inactive mutant effectively attenuated type I IFN induction. Collectively, our findings establish PCIF1 as a novel methyltransferase-independent suppressor of type I IFN responses, revealing its previously unrecognized non-catalytic function. This discovery offers critical insights into the multifaceted regulation of innate immunity and highlights PCIF1's non-catalytic function as a promising therapeutic target for modulating antiviral responses and inflammatory diseases.

Keywords: IRF3; PCIF1; antiviral response; innate immunity; m6Am; mRNA modifications; transcriptional regulation; type I interferon.

MeSH terms

  • Animals
  • HEK293 Cells
  • Humans
  • Immunity, Innate
  • Interferon Regulatory Factor-3* / metabolism
  • Interferon Type I* / metabolism
  • Methyltransferases* / metabolism
  • Mice
  • Phosphorylation
  • Poly I-C / pharmacology
  • STAT1 Transcription Factor / metabolism

Substances

  • Interferon Regulatory Factor-3
  • Interferon Type I
  • Methyltransferases
  • IRF3 protein, human
  • STAT1 Transcription Factor
  • Poly I-C