Targeting Mast Cells in Chronic Spontaneous Urticaria

Curr Allergy Asthma Rep. 2026 Feb 16;26(1):9. doi: 10.1007/s11882-025-01245-2.

Abstract

Purpose of review: This review focuses on the pathophysiology, diagnostic approach, and current and emerging treatments of chronic spontaneous urticaria (CSU), with an emphasis on mast-cell mediated mechanisms and therapeutic targets.

Recent findings: CSU is a mast-cell mediated disease involving both immunoglobulin E (IgE) and non-IgE mediated pathways, thus targeting mast cells and their downstream mediators can provide therapeutic benefit. Emerging therapies such as dupilumab, Bruton's tyrosine kinase (BTK) inhibitors, anti-KIT antibodies, Janus kinase (JAK) inhibitors, Mas-related G protein-coupled receptor X2 (MRGPRX2) inhibitors, interleukin (IL)-17 and IL-5 inhibitors, anti-thymic stromal lymphopoietin (TSLP) monoclonal antibodies, and mast cell silencers, as well as lifestyle changes such as low-histamine diets, are under investigation for antihistamine- refractory disease. While current international guidelines recommend second-generation H1-antihistamines as first-line treatments of CSU, novel treatments targeting mast-cell mediated pathways show promise for refractory disease. Recent advancements in targeted therapies and biomarkers may improve treatment personalization and response.

Keywords: Chronic Spontaneous Urticaria; Mast Cell; Novel Treatment.

Publication types

  • Review

MeSH terms

  • Animals
  • Chronic Urticaria* / diagnosis
  • Chronic Urticaria* / drug therapy
  • Chronic Urticaria* / immunology
  • Chronic Urticaria* / therapy
  • Humans
  • Mast Cells* / drug effects
  • Mast Cells* / immunology
  • Molecular Targeted Therapy