Lipopolysaccharide-targeting treatments for multidrug-resistant Pseudomonas aeruginosa

Expert Opin Ther Targets. 2026 Mar;30(3):203-211. doi: 10.1080/14728222.2026.2639679. Epub 2026 Mar 5.

Abstract

Introduction: Pseudomonas aeruginosa is an opportunistic, nosocomial, Gram-negative pathogen implicated in a wide variety of infection types and is especially problematic in chronic lung infections for patients with cystic fibrosis. Resistance to current antibiotics is frequent and rising, posing a serious public health threat, so development of new treatments is urgent.

Areas covered: This review aims to describe the current variety of LPS-targeting anti-Pseudomonals, including antimicrobials, bacteriophages, and pyocins, and how research is working to combat the rise of multi-drug resistant (MDR) P. aeruginosa infections.

Expert opinion: Pyocins, bacteriocins produced by P. aeruginosa, are an attractive potential treatment for MDR infections. Their high species-specificity, effective bactericidal activity, and relative stability and safety give them a promising treatment profile. It is likely that pyocin treatments could enter clinical testing, offering another lifeline for the future of combating P. aeruginosa.

Keywords: Antimicrobials; Pseudomonas aeruginosa; lipopolysaccharide; multi-drug resistance; phage therapy; pyocins.

Publication types

  • Review

MeSH terms

  • Animals
  • Anti-Bacterial Agents* / adverse effects
  • Anti-Bacterial Agents* / pharmacology
  • Cystic Fibrosis / complications
  • Cystic Fibrosis / microbiology
  • Drug Resistance, Multiple, Bacterial
  • Humans
  • Lipopolysaccharides / metabolism
  • Pseudomonas Infections* / drug therapy
  • Pseudomonas Infections* / microbiology
  • Pseudomonas aeruginosa* / drug effects
  • Pseudomonas aeruginosa* / isolation & purification
  • Pyocins / pharmacology
  • Species Specificity

Substances

  • Anti-Bacterial Agents
  • Lipopolysaccharides
  • Pyocins