Fisetin alleviates lipopolysaccharide-induced mastitis by inhibiting ferroptosis and modulating the gut microbiota

Vet Q. 2026 Dec;46(1):2642789. doi: 10.1080/01652176.2026.2642789. Epub 2026 Mar 17.

Abstract

Bovine mastitis poses an enormous challenge to the dairy industry. At present, dependence on antibiotic therapy has led to problems such as antibiotic-resistant bacteria and drug residues. Therefore, it is very important to seek alternative therapies for the treatment of bovine mastitis. Fisetin (FIS) with antioxidant and anti-inflammatory properties is found in various fruits and vegetables, although its regulatory role in mastitis treatment remains unclear. In the present study, we employed lipopolysaccharide (LPS)-induced cellular and animal mastitis models to investigate the regulatory effects of FIS on oxidative stress and ferroptosis pathways in mastitis treatment, utilizing techniques such as western blot, quantitative real-time PCR (qRT-PCR), immunofluorescence, hematoxylin-eosin (HE) staining, ROS, MDA, SOD, T-AOC, tissue total iron content analysis, mouse gut microbiota sequencing, and untargeted metabolomics. The results demonstrated that FIS modulates oxidative stress and ferroptosis pathways, leading to a reduction in intracellular and mouse mammary tissue inflammatory cytokines level. Furthermore, FIS treatment altered the gut microbiota structure and metabolites in LPS-induced mice, increasing short-chain fatty acid (SCFA) levels, which contributed to the restoration of the blood-milk barrier and alleviation of mastitis. This study could lead to novel therapeutic strategies for bovine mastitis based on traditional Chinese medicine.

Keywords: Bovine mastitis; Ferroptosis; Fisetin; Gut metabolites; Gut microbiota; Oxidative stress.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / pharmacology
  • Antioxidants / pharmacology
  • Cattle
  • Female
  • Ferroptosis* / drug effects
  • Flavonoids* / pharmacology
  • Flavonols* / pharmacology
  • Gastrointestinal Microbiome* / drug effects
  • Lipopolysaccharides
  • Mastitis* / chemically induced
  • Mastitis* / drug therapy
  • Mastitis, Bovine* / chemically induced
  • Mastitis, Bovine* / drug therapy
  • Mice
  • Mice, Inbred BALB C
  • Oxidative Stress / drug effects

Substances

  • Lipopolysaccharides
  • Flavonols
  • fisetin
  • Anti-Inflammatory Agents
  • Antioxidants
  • Flavonoids