Biomineralized nanoemulsion delivers mRNA for potent cancer immunotherapy

J Control Release. 2026 Jun 10:394:114889. doi: 10.1016/j.jconrel.2026.114889. Epub 2026 Mar 31.

Abstract

mRNA vaccines show great promise in cancer immunotherapy by eliciting potent cellular immune responses. Lipid nanoparticles (LNPs), validated through widespread use in COVID-19 vaccination, have become the most widely studied platform. However, their reliance on PEGylated lipids and tendency for hepatic accumulation may pose limitations for broader applications. To address these concerns, we developed a PEG-free nanoemulsion (NE) platform to deliver mRNA and minimize hepatic accumulation. We further employed a biomineralization strategy to anchor Mn2+ onto human serum albumin (HSA), thereby mitigating the cytotoxicity of free Mn2+ and forming a manganese-modified nanoemulsion (MnNE), which effectively activates the STING pathway. Compared with the LNP formulation of Moderna, MnNE showed superior transfection efficiency in antigen-presenting cells (APCs) following intramuscular injection. Using ovalbumin (OVA) as a model antigen, MnNE-mOVA elicited strong antigen-specific humoral and cellular immune responses. In both prophylactic and therapeutic E.G7-OVA tumor models, MnNE-mOVA significantly suppressed tumor growth and prolonged the survival compared with LNP-based formulations. Also, among all treatment groups, MnNE-mOVA most effectively reversed the immunosuppressive tumor microenvironment. These findings demonstrated that MnNE represented a safe and effective mRNA vaccine platform with substantial potential for cancer immunotherapy.

Keywords: Antitumor immunotherapy; Nanoemulsion; mRNA vaccine.

MeSH terms

  • Animals
  • Cancer Vaccines* / administration & dosage
  • Cell Line, Tumor
  • Emulsions
  • Female
  • Humans
  • Immunotherapy* / methods
  • Mice
  • Mice, Inbred C57BL
  • Nanoparticles* / administration & dosage
  • Nanoparticles* / chemistry
  • Neoplasms* / immunology
  • Neoplasms* / therapy
  • Ovalbumin / immunology
  • RNA, Messenger* / administration & dosage
  • Serum Albumin, Human / chemistry
  • mRNA Vaccines* / administration & dosage

Substances

  • Emulsions
  • Ovalbumin
  • RNA, Messenger
  • Cancer Vaccines
  • Serum Albumin, Human
  • mRNA Vaccines