Orai1 Facilitates Angiogenesis After Myocardial Infarction Through Notch1 Signaling Pathway

Arterioscler Thromb Vasc Biol. 2026 Jun;46(6):e324231. doi: 10.1161/ATVBAHA.125.324231. Epub 2026 Apr 16.

Abstract

Background: Post-ischemic neovascularization is crucial for cardiac repair after myocardial infarction (MI). While Orai1-dependent store-operated calcium entry is known to support angiogenesis, its specific role after MI remains unclear.

Methods: We stimulated human umbilical vein endothelial cells (ECs) with serum from patients with ST-segment-elevation MI to analyze proangiogenic mechanisms and to mimic the post-infarct systemic environment. We performed integrative analysis, including transcriptomics, proteomics, post-MI mouse heart single-cell RNA sequencing, and immunostaining.

Results: ST-segment-elevation MI serum enhanced angiogenesis by upregulating VEGF (vascular endothelial growth factor), Notch, and Ca2+ signaling pathways in EC. Notably, it increased Orai1 expression and store-operated calcium entry activity, required for EC migration and proliferation. Consistently, Orai1 inhibition with CM4620 significantly impaired subintestinal venous plexus development in zebrafish embryos. Single-cell RNA sequencing confirmed Orai1 upregulation, particularly in tip cells and proliferating EC clusters, which was confirmed in peri-infarct regions of mouse hearts and in tip-like cells in a 3-dimensional culture model. Proteomics analysis revealed that Orai1 silencing dysregulated VEGF and Notch1-related proangiogenic proteins. Furthermore, IL (interleukin)-17A mimicked ST-segment-elevation MI serum, inducing Orai1-mediated store-operated calcium entry and EC migration.

Conclusions: Together, these findings reveal a novel role for the Orai1-dependent mechanism in post-MI angiogenesis, highlighting Orai1 as a potential therapeutic target for cardiac repair.

Keywords: angiogenesis; coronary vessels; endothelial cells; interleukin-17; myocardial infarction.

MeSH terms

  • Angiogenesis
  • Animals
  • Calcium Signaling
  • Cell Movement
  • Cell Proliferation
  • Disease Models, Animal
  • Female
  • Human Umbilical Vein Endothelial Cells / metabolism
  • Humans
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Neovascularization, Physiologic*
  • ORAI1 Protein* / genetics
  • ORAI1 Protein* / metabolism
  • Receptor, Notch1* / genetics
  • Receptor, Notch1* / metabolism
  • ST Elevation Myocardial Infarction* / genetics
  • ST Elevation Myocardial Infarction* / metabolism
  • ST Elevation Myocardial Infarction* / pathology
  • ST Elevation Myocardial Infarction* / physiopathology
  • Signal Transduction
  • Vascular Endothelial Growth Factor A / genetics
  • Vascular Endothelial Growth Factor A / metabolism
  • Zebrafish

Substances

  • ORAI1 Protein
  • Receptor, Notch1
  • ORAI1 protein, human
  • NOTCH1 protein, human
  • Vascular Endothelial Growth Factor A
  • Orai1 protein, mouse
  • Notch1 protein, mouse
  • VEGFA protein, human