Competitive inhibition of drug-protein interaction in eye fluids and tissues

J Pharm Sci. 1973 Dec;62(12):1942-5. doi: 10.1002/jps.2600621207.
No abstract available

MeSH terms

  • Animals
  • Binding, Competitive
  • Biopharmaceutics
  • Cetylpyridinium / pharmacology
  • Cornea / drug effects
  • Dialysis
  • Dose-Response Relationship, Drug
  • Drug Antagonism
  • Ethylenediamines / metabolism
  • Eye / metabolism*
  • Eye Proteins / metabolism*
  • In Vitro Techniques
  • Male
  • Methylprednisolone / metabolism
  • Miotics / pharmacology
  • Naphthalenes / metabolism
  • Pharmaceutical Preparations / metabolism*
  • Pilocarpine / pharmacology
  • Protein Binding / drug effects
  • Rabbits
  • Serum Albumin / metabolism
  • Sulfisoxazole / metabolism
  • Surface-Active Agents / pharmacology
  • Time Factors

Substances

  • Ethylenediamines
  • Eye Proteins
  • Miotics
  • Naphthalenes
  • Pharmaceutical Preparations
  • Serum Albumin
  • Surface-Active Agents
  • Pilocarpine
  • Sulfisoxazole
  • Cetylpyridinium
  • Methylprednisolone