Brain arylamidase. Purfication and characterization of the soluble bovine enzyme

Biochem J. 1969 Apr;112(3):335-42. doi: 10.1042/bj1120335.

Abstract

1. An enzyme acting on aminoacyl-beta-naphthylamides has been isolated from the soluble fraction of bovine brain and purified 205-fold by means of ammonium sulphate fractionation, hydroxyapatite adsorption and DEAE-Sephadex column chromatography. 2. Arylamidase requires thiol groups for retention of its activity, is heat-labile and is susceptible to freezing. p-Chloromercuribenzoate and N-ethylmaleimide inactivate the enzyme rapidly. 3. Metal ions are not required for its activity, but stimulation by Mn(2+) and Mg(2+) and inactivation by Co(2+) and Zn(2+) are observed. 4. Optimum pH7.5 in phosphate buffer was exhibited for all substrates tested except l-leucyl-beta-naphthylamide, for which optimum pH is 6.5. 5. K(m) values for a number of substrates have been obtained and substrate inhibition at high concentrations was demonstrated. 6. The molecular weight is approx. 70000 as determined by Sephadex-gel filtration.

MeSH terms

  • Aminopeptidases* / isolation & purification
  • Animals
  • Brain / enzymology*
  • Cattle
  • Chemical Phenomena
  • Chemical Precipitation
  • Chemistry
  • Chloromercuribenzoates
  • Chromatography, Gel
  • Chromatography, Ion Exchange
  • Cobalt
  • Electrophoresis, Disc
  • Ethylmaleimide
  • Freezing
  • Hot Temperature
  • Hydrogen-Ion Concentration
  • Hydroxyapatites
  • Kinetics
  • Magnesium
  • Manganese
  • Methods
  • Molecular Weight
  • Naphthalenes
  • Quaternary Ammonium Compounds
  • Solubility
  • Sulfhydryl Compounds
  • Zinc

Substances

  • Chloromercuribenzoates
  • Hydroxyapatites
  • Naphthalenes
  • Quaternary Ammonium Compounds
  • Sulfhydryl Compounds
  • Cobalt
  • Manganese
  • Aminopeptidases
  • Magnesium
  • Zinc
  • Ethylmaleimide