Demonstration of adenosine receptors on mouse cerebral smooth muscle membranes

Stroke. 1984 Jul-Aug;15(4):725-7. doi: 10.1161/01.str.15.4.725.

Abstract

Adenosine receptors have been identified on brain cortical membranes and microvascular preparations. However, they have not been demonstrated on specific microvascular elements in isolation. 2-3H-chloroadenosine was used as a ligand to investigate the presence of adenosine receptors on isolated mouse cerebral smooth muscle membranes. The binding studies reveal the presence of a high affinity binding site with a Kd value of 33.3 nM and a maximal binding capacity (Bmax) of 283 fmol/mg protein. These findings demonstrate that there is an adenosine receptor on cerebral smooth muscle membranes.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 2-Chloroadenosine
  • Adenosine / analogs & derivatives
  • Adenosine / metabolism
  • Animals
  • Brain / blood supply*
  • Cell Membrane / analysis
  • In Vitro Techniques
  • Mice
  • Microcirculation
  • Muscle, Smooth, Vascular / analysis*
  • Receptors, Cell Surface / analysis*
  • Receptors, Cell Surface / metabolism
  • Receptors, Purinergic
  • Tritium

Substances

  • Receptors, Cell Surface
  • Receptors, Purinergic
  • Tritium
  • 2-Chloroadenosine
  • Adenosine