The anticalmodulin drugs trifluoperazine and R24571 remove the activation of the purified erythrocyte Ca2+-ATPase by acidic phospholipids and by controlled proteolysis

FEBS Lett. 1982 Jun 21;143(1):65-8. doi: 10.1016/0014-5793(82)80274-3.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calcium-Binding Proteins / antagonists & inhibitors*
  • Calcium-Transporting ATPases / blood*
  • Calmodulin / antagonists & inhibitors*
  • Enzyme Activation
  • Erythrocyte Membrane / enzymology*
  • Erythrocytes / enzymology*
  • Humans
  • Imidazoles / pharmacology*
  • Kinetics
  • Phosphatidylcholines
  • Phospholipids / pharmacology*
  • Trifluoperazine / pharmacology*

Substances

  • Calcium-Binding Proteins
  • Calmodulin
  • Imidazoles
  • Phosphatidylcholines
  • Phospholipids
  • Trifluoperazine
  • calmidazolium
  • asolectin
  • Calcium-Transporting ATPases