Dephosphorylation of synthetic phosphopeptides by protein phosphatase-T, a phosphothreonyl protein phosphatase

J Biol Chem. 1982 Aug 10;257(15):8565-8.

Abstract

The synthetic phosphohexapeptides Arg-Arg-Ala-Thr(35P)-Val-Ala and Arg-Arg-Ala-Ser(32P)-Val-Ala, phosphorylated by the cAMP-dependent protein kinase and differing only in the nature of the phosphorylated residue, have been used as substrates of a partially purified rat liver protein phosphatase-T, distinct from the multifunctional protein phosphatase-1. While the phosphothreonyl hexapeptide is readily dephosphorylated (exhibiting a Km = 15 microM), the phosphoseryl one is almost unaffected. Such a behavior is not shared by protein phosphatase-1, calf intestine alkaline phosphatase, and potato acid phosphatase, all of which are more active on the phosphoseryl hexapeptide. The NH2-terminal basic residues critical for cAMP-dependent phosphorylation are not required in the dephosphorylation reaction, as both Arg can be removed without impairing the efficiency of protein phosphatase-T toward the phosphothreonyl peptide. On the other hand, the replacement of 2 Pro for the Ala and Val flanking Thr(32P), to give a new phosphohexapeptide reproducing the phosphorylated site of protein phosphatase inhibitor-1, prevents the protein phosphatase-T activity. Moreover, IgG heavy chain 32P labeled in tyrosine is not affected by protein phosphatase-T, while it is dephosphorylated by alkaline phosphatase. These results would indicate that protein phosphatase(s)-T represent a distinct class of protein phosphatases specifically involved in the dephosphorylation of phosphothreonyl residues fulfilling definite structural requirements.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acid Phosphatase / metabolism
  • Alkaline Phosphatase / metabolism
  • Amino Acid Sequence
  • Animals
  • Cyclic AMP / metabolism
  • Kinetics
  • Oligopeptides / metabolism
  • Phosphopeptides / metabolism*
  • Phosphoprotein Phosphatases / metabolism*
  • Phosphorylase Phosphatase / metabolism
  • Phosphorylation
  • Phosphothreonine / metabolism
  • Protein Kinases / metabolism
  • Protein Phosphatase 1
  • Rats

Substances

  • Oligopeptides
  • Phosphopeptides
  • Phosphothreonine
  • Cyclic AMP
  • Protein Kinases
  • protein phosphatase-T
  • Alkaline Phosphatase
  • Phosphoprotein Phosphatases
  • Protein Phosphatase 1
  • Phosphorylase Phosphatase
  • Acid Phosphatase