Regulation of the strength of adenosine modulation in the hippocampus by a differential distribution of the density of A1 receptors

Brain Res. 1983 Jan 31;260(1):156-9. doi: 10.1016/0006-8993(83)90779-5.

Abstract

Correlative studies examining: (1) the binding of [3H]cyclohexyladenosine to A1 adenosine receptor sites, and (2) the depressive action of adenosine on evoked activity, were performed in the hippocampal formation. A greater number of A1 sites was observed in the dorsal versus ventral aspect of the hippocampus, and a larger depression of evoked potentials by adenosine was obtained in the dorsal aspect. These observations suggest that a differential density of A1 receptors might control the magnitude of modulatory action by adenosine on hippocampal circuitry.

MeSH terms

  • Adenosine / analogs & derivatives
  • Adenosine / metabolism
  • Adenosine / pharmacology*
  • Animals
  • Culture Techniques
  • Evoked Potentials / drug effects
  • Hippocampus / drug effects*
  • Male
  • Rats
  • Receptors, Cell Surface / drug effects*
  • Receptors, Purinergic
  • Synaptic Transmission / drug effects*

Substances

  • Receptors, Cell Surface
  • Receptors, Purinergic
  • N(6)-cyclohexyladenosine
  • Adenosine