Effect on neuronal and non-neuronal benzodiazepine binding sites

Neurochem Res. 1983 Sep;8(9):1135-41. doi: 10.1007/BF00964927.

Abstract

The frontal cortex, hippocampus, and cerebellum of the Fischer 344 rat were examined for an age-dependent change in neuronal and non-neuronal binding. Clonazepam and Ro5-6669 displaceable [3H]diazepam binding were used as indicators of [3H]diazepam binding on neuronal and non-neuronal membranes, respectively. In both the frontal cortex and the hippocampus, clonazepam displaceable [3H]diazepam binding in the senescent rat was significantly less than the young and mature rat. In the frontal cortex, Ro5-6669 did not significantly displace [3H]diazepam binding in any age group. The Ro5-6669 displaceable [3H]diazepam binding in the hippocampus was not altered with age. In the cerebellum clonazepam and Ro5-6669 displaceable binding in the old rat was significantly less and more, respectively, compared to the young rat.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Aging*
  • Animals
  • Benzodiazepines / metabolism*
  • Benzodiazepinones
  • Binding Sites
  • Cerebellum / metabolism
  • Clonazepam / metabolism
  • Frontal Lobe / metabolism
  • Hippocampus / metabolism
  • Male
  • Neurons / metabolism*
  • Rats
  • Rats, Inbred F344

Substances

  • Benzodiazepinones
  • Benzodiazepines
  • Clonazepam
  • Ro 5-6669