Effect of a perfluorocarbon emulsion (Fluosol-DA) on reticuloendothelial system clearance function

Am J Hematol. 1984 Jan;16(1):15-21. doi: 10.1002/ajh.2830160103.

Abstract

To study the effect of a perfluorocarbon oxygen transport emulsion (Fluosol-DA) on reticuloendothelial system (RES) function, we measured the blood clearance of human erythrocytes transfused to rats. Compared with saline treatment, Fluosol-DA at 30 ml/kg doses significantly increased both the percent 20-hour blood recovery (mean 8.9% +/- 2.7 SEM vs 1.3% +/- 0.25 SEM) and 51Cr t1/2 survival (mean 14.0 hours +/- 2.7 SEM vs 3.5 hours +/- 0.33 SEM) of the human red cells. This suppression of RES clearance function was transient and no longer detectable seven days after single Fluosol-DA doses. The Fluosol-DA-induced RES block was about three times greater than that obtainable with 4 g/kg of a soybean oil emulsion used for clinical hyperalimentation. On the other hand, the effect of ethyl palmitate (0.5 g/kg), a potent but toxic RES blocker, was 3.5 times greater than that of Fluosol-DA in this test system. If Fluosol-DA also induces RES block in humans, this emulsion could be explored as a therapeutic RES blocker in certain immune cytopenias.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Dose-Response Relationship, Drug
  • Drug Combinations / pharmacology
  • Fluorocarbons / pharmacology*
  • Half-Life
  • Hydroxyethyl Starch Derivatives
  • Kinetics
  • Male
  • Mononuclear Phagocyte System / drug effects
  • Mononuclear Phagocyte System / physiology*
  • Phagocytosis
  • Rats
  • Rats, Inbred Strains

Substances

  • Drug Combinations
  • Fluorocarbons
  • Hydroxyethyl Starch Derivatives
  • glucose, glycerol, hydroxyethyl starch, perfluorodecalin, perfluorotripropylamine, pluronic F-68, salts, yolk phospholipids drug combination