8-Azaguanine versus 6-thioguanine: influence on frequency and expression time of induced HGPRT- mutations in Chinese hamster V79 cells

Mutat Res. 1983 Feb;107(2):397-411. doi: 10.1016/0027-5107(83)90179-3.

Abstract

Chinese hamster V79 cells were mutagenized with ethyl methanesulfonate at various concentrations. Clones resistant to 8-azaguanine (20 and 80 micrograms/ml) or 6-thioguanine (4 micrograms/ml) were selected at different times after the treatments. The total yield of induced mutations was only slightly affected by the kind and concentration of purine analog used in the selection. However, full phenotypic expression of the mutants selected with 8-azaguanine was achieved earlier than that of mutants resistant to 6-thioguanine. This result seems to be best explained by the reported lower affinity of 8-azaguanine for the wild-type HGPRT enzyme, thus providing evidence that, in this gene-mutation assay, the phenotypic expression time has a physiological component.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Azaguanine / pharmacology*
  • Cell Survival / drug effects
  • Clone Cells / drug effects
  • Cricetinae
  • Cricetulus
  • Drug Resistance
  • Ethyl Methanesulfonate / pharmacology
  • Hypoxanthine Phosphoribosyltransferase / genetics*
  • Mutation*
  • Phenotype
  • Thioguanine / pharmacology*
  • Time Factors

Substances

  • Ethyl Methanesulfonate
  • Hypoxanthine Phosphoribosyltransferase
  • Thioguanine
  • Azaguanine