Structure and function of an acetylcholine receptor

Biophys J. 1982 Jan;37(1):371-83. doi: 10.1016/S0006-3495(82)84685-7.

Abstract

Structural analysis of an acetylcholine receptor from Torpedo californica leads to a three-dimensional model in which a "monomeric" receptor is shown to contain subunits arranged around a central ionophoretic channel, which in turn traverses the entire 110 A length of the molecule. The receptor extends approximately 15 A on the cytoplasmic side, 55 A on the synaptic side of the membrane. The alpha-bungarotoxin/agonist binding site is found to be approximately 55 A from the entrance to the central gated ion channel. A hypothesis for the mechanism of AcChR is presented which takes into account the structural and kinetic data, which is testable, and which serves as a focus for future studies on the agonist-induced structure change in AcChR.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Bungarotoxins / pharmacology
  • Models, Biological
  • Molecular Conformation
  • Neurotoxins / pharmacology*
  • Receptors, Cholinergic / drug effects
  • Receptors, Cholinergic / isolation & purification
  • Receptors, Cholinergic / ultrastructure*
  • Torpedo

Substances

  • Bungarotoxins
  • Neurotoxins
  • Receptors, Cholinergic