Imaging the primate adrenal medulla with [123I] and [131I] meta-iodobenzylguanidine: concise communication

J Nucl Med. 1981 Apr;22(4):358-64.

Abstract

An evaluation of radioiodinated meta-iodobenzylguanidine (m-IBG) as an adrenomedullary imaging agent is reported in 15 rhesus monkeys. Scintiscans of the monkey adrenal medulla have been obtained with [123I]- and [m-131I]IBG at 2-6 days after injection. The imaging superiority of m-IBG over its positional isomer, para-iodobenzylguanidine (p-IBG), is documented in both dogs and monkeys. Administration of reserpine, a depletor of catecholamine stores, markedly lowers the [m-131I]-IBG content of the dog adrenal medulla, but the adrenergic blocking agents phenoxybenzamine and propranolol have no effect. Subcellular fractionation of the dog's adrenal medullae reveals that m-IBG is sequestered mainly in the chromaffin storage granules. The results of this study suggest that radioiodinated m-IBG, previously reported to image the primate myocardium, also merits evaluation as a clinical radiopharmaceutical for the adrenal medulla.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 3-Iodobenzylguanidine
  • Adrenal Medulla / diagnostic imaging*
  • Adrenal Medulla / metabolism
  • Adrenal Medulla / ultrastructure
  • Animals
  • Chromaffin Granules / metabolism
  • Dogs
  • Female
  • Guanidines* / metabolism
  • Iodine Radioisotopes*
  • Iodobenzenes*
  • Macaca mulatta
  • Male
  • Radionuclide Imaging
  • Reserpine / pharmacology
  • Tissue Distribution

Substances

  • Guanidines
  • Iodine Radioisotopes
  • Iodobenzenes
  • 4-iodobenzylguanidine
  • 3-Iodobenzylguanidine
  • Reserpine