Behavioural assessment in rats of the antipsychotic potential of the potent dopamine D2 receptor antagonist, (-)eticlopride

Pharmacol Res. 1995 May;31(5):261-7. doi: 10.1016/1043-6618(95)80030-1.

Abstract

The effects of the selective D2 DA receptor antagonist, (-)eticlopride, a drug belonging to the benzamide class, were investigated on the D2 DA agonist SND 919- and CQP 201-403-induced stereotyped behaviour and on CQP 201-403-induced shaking, in rats, and on isolation-induced aggression, in mice. (-)Eticlopride was also tested over a wide dose range (5-1200 micrograms kg-1, s.c.) for sedative and cataleptic activity, in rats. For comparison, some experiments were performed with (-)sulpiride (10 and 40 mg kg-1, s.c.) The data obtained show that (-)eticlopride differs from (-)sulpiride and potentially modifies animal behaviour, whether spontaneous or induced; moreover, they suggest a potential clinical use for this neuroleptic in the management of psychotic states.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aggression / drug effects
  • Animals
  • Antipsychotic Agents / pharmacology
  • Behavior, Animal / drug effects*
  • Dopamine D2 Receptor Antagonists*
  • Male
  • Mice
  • Mice, Inbred Strains
  • Motor Activity / drug effects*
  • Rats
  • Rats, Inbred Strains
  • Salicylamides / pharmacology*
  • Stereotyped Behavior / drug effects*
  • Sulpiride / pharmacology

Substances

  • Antipsychotic Agents
  • Dopamine D2 Receptor Antagonists
  • Salicylamides
  • Sulpiride
  • eticlopride