Stoichiometry of a recombinant GABAA receptor deduced from mutation-induced rectification

Neuroreport. 1993 Dec 13;5(3):285-8. doi: 10.1097/00001756-199312000-00026.

Abstract

Ligand-gated ion channels generally display a heterooligomeric subunit structure. The present report describes an electrophysiological method that provides criteria indicating the subunit stoichiometry of a recombinant GABAA receptor composed of alpha 3, beta 2 and gamma 2 subunits. Our results exclude the stoichiometries 3 alpha 1 beta 1 gamma, 1 alpha 3 beta 1 gamma, 1 alpha 1 beta 3 gamma and suggest that the possible subunit stoichiometries for this receptor are 2 alpha 1 beta 2 gamma, 2 alpha 2 beta 1 gamma or 1 alpha 2 beta 2 gamma, of which the alpha subunit composition 2 alpha 1 beta 2 gamma may be favoured. The method is based on the quantification of the outward rectification of the GABA-evoked current induced by point mutation of charged amino acids located near the ion channel pore.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Cell Line
  • Electrophysiology
  • Humans
  • Ion Channels / metabolism
  • Kidney / cytology
  • Kidney / metabolism
  • Molecular Sequence Data
  • Mutation*
  • Rats
  • Receptors, GABA-A / genetics*
  • Recombinant Proteins / genetics

Substances

  • Ion Channels
  • Receptors, GABA-A
  • Recombinant Proteins