Selectivity of connexin-specific gap junctions does not correlate with channel conductance

Circ Res. 1995 Dec;77(6):1156-65. doi: 10.1161/01.res.77.6.1156.

Abstract

Connexins form a variety of gap junction channels that vary in their developmental and tissue-specific levels of expression, modulation of gating by transjunctional voltage and posttranslational modification, and unitary channel conductance (gamma j). Despite a 10-fold variation in gamma j, whether connexin-specific channels possess distinct ionic and molecular permeabilities is presently unknown. A major assumption of the conventional model for a gap junction channel pore is that gamma j is determined primarily by pore diameter. Hence, molecular size permeability limits should increase and ionic selectivity should decrease with increasing channel gamma j (and pore diameter). Equimolar ion substitution of 120 mmol/L KCl for potassium glutamate was used to determine the unitary conductance ratios for rat connexin40 and connexin43, chicken connexin43 and connexin45, and human connexin37 channels functionally expressed in communication-deficient mouse neuroblastoma (N2A) cells. Comparison of experimental and predicted conductance ratios based on the aqueous mobilities of all ions according to the Goldman-Hodgkin-Katz current equation was used to determine relative anion-to-cation permeability ratios. Direct correlation of junctional conductance with dye transfer of two fluorescein-derivatives (2 mmol/L 6-carboxyfluorescein or 2',7'-dichlorofluorescein) was also performed. Both approaches revealed a range of selectivities and permeabilities for all five different connexins that was independent of channel conductance. These results are not consistent with the conventional simple aqueous pore model of a gap junction channel and suggest a new model for connexin channel conductance and permselectivity based on electrostatic interactions. Divergent conductance and permeability properties are features of other classes of ion channels (eg, Na+ and K+ channels), implying similar mechanisms for selectivity.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Blotting, Northern
  • Cells, Cultured
  • Chickens
  • Connexins / genetics
  • Connexins / metabolism*
  • Diffusion
  • Electric Conductivity
  • Electrophysiology
  • Fluoresceins
  • Fluorescent Dyes
  • Gap Junctions / metabolism*
  • Gap Junctions / physiology
  • Genetic Vectors
  • Humans
  • Ion Channels / genetics
  • Ion Channels / metabolism*
  • Ion Channels / physiology
  • Liposomes
  • Mice
  • Models, Anatomic
  • Models, Biological
  • Molecular Weight
  • Neuroblastoma
  • Patch-Clamp Techniques
  • Phosphatidylethanolamines
  • Plasmids / genetics
  • Rats
  • Second Messenger Systems
  • Surface Properties
  • Transfection

Substances

  • Connexins
  • Fluoresceins
  • Fluorescent Dyes
  • Ion Channels
  • Liposomes
  • Phosphatidylethanolamines
  • 6-carboxyfluorescein
  • 2',7'-dichlorofluorescein
  • 1,2-dielaidoylphosphatidylethanolamine