Topoisomerase poisons: harnessing the dark side of enzyme mechanism

J Biol Chem. 1995 Sep 15;270(37):21429-32. doi: 10.1074/jbc.270.37.21429.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.
  • Review

MeSH terms

  • Animals
  • Bacteria / enzymology
  • Cell Death
  • DNA / chemistry
  • DNA / metabolism
  • DNA Replication
  • DNA Topoisomerases, Type I / metabolism*
  • DNA Topoisomerases, Type II / metabolism*
  • Enzyme Inhibitors / pharmacology*
  • Enzyme Inhibitors / toxicity
  • Topoisomerase I Inhibitors
  • Topoisomerase II Inhibitors

Substances

  • Enzyme Inhibitors
  • Topoisomerase I Inhibitors
  • Topoisomerase II Inhibitors
  • DNA
  • DNA Topoisomerases, Type I
  • DNA Topoisomerases, Type II