Hydroxyl radical-scavenging property of indomethacin

Mol Cell Biochem. 1994 Jul 27;136(2):139-44. doi: 10.1007/BF00926074.

Abstract

The ability of indomethacin to scavenge hydroxyl radical (.OH) using high pressure liquid chromatography (HPLC) was investigated. .OH radical was generated by photolysis of H2O2 (1.5-10 mmoles/L) with UV light and was trapped with salicyclic acid (500 nmoles). H2O2 produced .OH in a concentration-dependent manner as estimated by .OH adduct products 2,3- and 2,5-dihydroxybenzoic acid (DHBA). Indomethacin in increasing concentrations (5-600 mumoles/L) produced increasing inhibition of generation of 2,3-DHBA (7-67%) and of 2,5-DHBA (7-77%). The results indicate that indomethacin scavenges .OH in a concentration-dependent manner.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Chromatography, High Pressure Liquid
  • Free Radical Scavengers / pharmacology*
  • Gentisates*
  • Hydroxybenzoates
  • Hydroxyl Radical
  • Indomethacin / pharmacology*
  • Photolysis
  • Sensitivity and Specificity
  • Ultraviolet Rays

Substances

  • Free Radical Scavengers
  • Gentisates
  • Hydroxybenzoates
  • Hydroxyl Radical
  • 2,3-dihydroxybenzoic acid
  • 2,5-dihydroxybenzoic acid
  • Indomethacin