Epileptiform activity induced by 4-aminopyridine in guinea-pig and rat neocortices

Neurosci Lett. 1993 May 14;154(1-2):157-60. doi: 10.1016/0304-3940(93)90195-q.

Abstract

Extracellular field recordings were performed in guinea-pig and rat neocortical slice preparations maintained in vitro. Bath application of the convulsant drug 4-aminopyridine (4-AP, 100 microM) induced spontaneous epileptiform potentials in 80% of the guinea-pig neocortical slices and only in 6% of the neocortical slices from rat. In both species spontaneous epileptiform activity consisted of a 4-16 s long ictal-like discharge that recurred with a frequency range of 0.01-0.02 Hz. In rat neocortical slices stimulus-induced responses resembled the spontaneous occurring epileptiform events. Ictal-like discharges in guinea-pig neocortical slices were blocked by the N-methyl-D-aspartate (NMDA) receptor antagonist 3-((+/-)-2-carboxypiperazine-4-yl)propyl-1-phosphonic acid (5 microM), while those in the rat disappeared during perfusion with the non-NMDA excitatory amino acid receptor antagonist 6-cyano-7-nitroquinoxaline-2,3-dione (1-3 microM). These results indicate that the neocortex of guinea-pig has a higher propensity to generate 4-AP-induced spontaneous epileptiform activity than that of rat. Furthermore the epileptiform activity in these two species requires a different involvement of excitatory amino acid receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 4-Aminopyridine*
  • 6-Cyano-7-nitroquinoxaline-2,3-dione
  • Animals
  • Anticonvulsants / pharmacology
  • Cerebral Cortex / drug effects
  • Cerebral Cortex / physiopathology*
  • Electric Stimulation
  • Electrophysiology
  • Epilepsy / chemically induced*
  • Epilepsy / physiopathology
  • Guinea Pigs
  • In Vitro Techniques
  • Piperazines / pharmacology
  • Quinoxalines / pharmacology
  • Rats
  • Receptors, N-Methyl-D-Aspartate / antagonists & inhibitors

Substances

  • Anticonvulsants
  • Piperazines
  • Quinoxalines
  • Receptors, N-Methyl-D-Aspartate
  • 6-Cyano-7-nitroquinoxaline-2,3-dione
  • 3-(2-carboxypiperazin-4-yl)propyl-1-phosphonic acid
  • 4-Aminopyridine