Modulation of the expression of murine lupus by gonadotropin-releasing hormone analogs

Endocrinology. 1994 Jun;134(6):2516-23. doi: 10.1210/endo.134.6.8194477.

Abstract

Recent studies have suggested that hypothalamic and pituitary hormones may directly influence the immune system. One such hormone with immunomodulatory properties is GnRH. We hypothesized that GnRH and/or the gonadotropins might alter the severity of autoimmune disease through mechanisms distinct from their effects on gonadal hormones. This possibility was tested in a murine model of lupus. We assessed disease severity over time in intact and castrated, male and female, lupus-prone (SWR x NZB) F1 hybrid mice during treatment with GnRH agonist, GnRH antagonist, or vehicle. Compared to vehicle administration, GnRH antagonist administration significantly decreased total serum immunoglobulin G and anti-DNA antibodies in castrated male and female mice and significantly improved survival. In contrast, GnRH agonist administration exerted reciprocal effects in castrated mice, leading to early increases in serum anti-DNA and total immunoglobulin G levels. We conclude that GnRH and/or the gonadotropins can modify the expression of murine lupus independently of their regulation of gonadal steroid secretion.

MeSH terms

  • Animals
  • Antibodies, Antinuclear / blood
  • Estradiol / pharmacology
  • Female
  • Flow Cytometry
  • Gonadotropin-Releasing Hormone / analogs & derivatives*
  • Gonadotropin-Releasing Hormone / antagonists & inhibitors
  • Gonadotropin-Releasing Hormone / therapeutic use*
  • Hematuria
  • Immunoglobulin G / blood
  • Lupus Erythematosus, Systemic / drug therapy*
  • Lupus Erythematosus, Systemic / immunology
  • Luteinizing Hormone / blood
  • Male
  • Mice
  • Mice, Mutant Strains
  • Oligopeptides / therapeutic use
  • Orchiectomy
  • Ovariectomy
  • Proteinuria

Substances

  • Antibodies, Antinuclear
  • Immunoglobulin G
  • LHRH, N-Ac-2-Nal(1)-4-Cl-Phe(2)-3-Pal(3)-Arg(5)-Glu(6)-AlaNH2(10)-
  • Oligopeptides
  • Gonadotropin-Releasing Hormone
  • Estradiol
  • Luteinizing Hormone
  • iturelix