An ion-sensitive microelectrode study on the effect of a high concentration of ivermectin on chloride balance in the somatic muscle bag cells of Ascaris suum

Parasitology. 1993 May:106 ( Pt 4):421-7. doi: 10.1017/s0031182000067172.

Abstract

Ivermectin has been shown to increase chloride conductances of invertebrate cells. On the muscle cells of the parasitic nematode Ascaris, ivermectin acts as both a GABA receptor antagonist and a chloride channel opener. In this study, ion-sensitive microelectrodes were used to investigate the effect of ivermectin on intracellular Cl- concentration of the somatic muscle bag cells of Ascaris suum. Incubation of muscle cells with ivermectin (10 microM in 1% dimethyl sulphoxide vehicle for 60 min) increased intracellular Cl- by 2.9 mM or 15% compared to controls (P < 0.01, n = 6).

MeSH terms

  • Animals
  • Ascaris suum / drug effects
  • Ascaris suum / physiology*
  • Chlorides / metabolism*
  • Dimethyl Sulfoxide / pharmacology
  • In Vitro Techniques
  • Ions
  • Ivermectin / pharmacology*
  • Membrane Potentials
  • Microelectrodes
  • Muscles / drug effects
  • Muscles / physiology*
  • Sensitivity and Specificity
  • Water-Electrolyte Balance / drug effects*

Substances

  • Chlorides
  • Ions
  • Ivermectin
  • Dimethyl Sulfoxide